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4-[(5-ethylpyridin-2-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-ethyl-N-[(3-fluorophenyl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
2-(3,3-dimethylbutanoyl)-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
ethyl 5-[5-(4-methoxyphenyl)furan-2-carbonyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-{[1-ethyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one
N-{2-[({3-hydroxy-1-[(3-methylphenyl)methyl]-2-oxopiperidin-3-yl}methyl)amino]ethyl}acetamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(1,3-benzothiazol-2-ylmethyl)-5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)pyrrolidin-2-one
5-fluoro-8-[6-(2-methoxyphenyl)pyridazin-3-yl]quinoline
5-(2,6-difluorophenoxymethyl)-N-[(3-methoxyphenyl)methyl]-1,2-oxazole-3-carboxamide
3-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
(3E)-N-(5-methyl-2-pentanamidophenyl)pent-3-enamide
(1S,5R)-6-(2-methoxyethyl)-3-[(5-phenylthiophen-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
methyl 3-[(3-ethoxyphenyl)methyl]-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
1-(3-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenyl)ethan-1-one
1-[3-(2-methylphenyl)benzoyl]-2-(pyrrolidine-1-carbonyl)piperazine
N-[2-(1H-imidazol-4-yl)ethyl]-4-propylpyrimidine-5-carboxamide
3-{3-[1-(morpholin-4-yl)ethyl]-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl}propanoic acid
4-methyl-6-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-N-(2-phenylethyl)piperidine-1-carboxamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[2-(oxan-2-yl)ethyl]benzamide
7-{[4-(2-methylpyridin-4-yl)piperazin-1-yl]methyl}-1H-indole
3-methyl-5-(2-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.4]nonan-7-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}[1-(thiophen-2-yl)ethyl]amine
5-(2H-1,3-benzodioxol-5-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,2,4-triazin-3-amine
2-(1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
N-(3,4-difluorophenyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
4-(5-methyl-2-phenylfuran-3-carbonyl)-1λ6-thiomorpholine-1,1-dione
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-(3-methoxypropyl)pyrimidine-5-carboxamide
7-chloro-4-(1,4-diazepan-1-yl)quinoline
2-[(2-ethylpyrimidin-5-yl)methyl]-7-(3-methylbenzoyl)-2,7-diazaspiro[4.5]decane
(2-{2-[2-(methoxymethyl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
3-(3-ethyl-1,2,4-oxadiazol-5-yl)-N,N-dimethylpiperidine-1-carboxamide
8-(1H-1,3-benzodiazole-5-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-cyclohexaneamido-1-(2-methoxyethyl)-N-[3-(methylsulfanyl)propyl]-1H-1,3-benzodiazole-7-carboxamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)(furan-2-ylmethyl)methylamine
1-{[3-(4-chlorophenoxy)phenyl]methyl}-4-methyl-1,4-diazepan-5-one
5-[3-(2-fluorophenyl)-1H-pyrazol-5-yl]-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
1-[2-(2-ethoxyphenyl)ethyl]-4-(1H-imidazol-2-yl)-1H-1,2,3-triazole
(3S,9aR)-8-(4-methylbenzoyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-(3-chlorophenyl)-4-[2-(pyrrolidin-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3R,5S)-5-(morpholine-4-carbonyl)-N-[2-(pyrazin-2-yl)ethyl]piperidine-3-carboxamide
3,5-difluoro-2-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
2-(4-fluoro-3-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)acetic acid
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-[2-(4-methoxyphenyl)ethyl]acetamide
1,3-dimethyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine