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5-chloro-2-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-3-methyl-1H-indole
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(4-methyl-1H-imidazole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-benzyl-N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-3-oxopiperazine-1-carboxamide
6-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,3-dimethyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
methyl 1-benzyl-3-cyclopropaneamido-5-{[(3-methoxyphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-methoxy-6-{[(2S,4R)-4-[(4-methoxyphenyl)sulfanyl]-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methyl}phenol
2-[(1-methyl-2,5-dioxo-2,3,4,5-tetrahydro-1H-1,4-benzodiazepin-4-yl)methyl]benzonitrile
8-(butan-2-yl)-1-methyl-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-(2-methylpropyl)-8-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
(1S,5R)-3-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-(pyridin-3-yl)-2-[4-(thiomorpholin-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]acetamide
2-(2-phenylethyl)-9-(propane-1-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-chlorophenyl)-4-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
1-[(4aS,8aS)-4a-hydroxy-7-(pyridin-4-ylmethyl)-decahydro-2,7-naphthyridin-2-yl]-3-ethoxypropan-1-one
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(4-methoxyphenoxy)piperidine
(3aR,5R,6S,7aS)-2-(3-methyl-1-benzothiophene-2-carbonyl)-octahydro-1H-isoindole-5,6-diol
(3R,9aR)-8-[(5-methylthiophen-2-yl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}-N-(pyridin-2-ylmethyl)acetamide
N-ethyl-N-[2-(3-methoxyphenoxy)ethyl]-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
3-chloro-4-fluoro-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-1-benzothiophene-2-carboxamide
3-(4-methoxyphenyl)-5-[(2-propyl-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
2-methyl-1-{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}-1,4-diazepan-5-one
1-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(2-fluorophenyl)methyl]piperidine
ethyl 4-[(2-chlorophenyl)methyl]-1-[(3-hydroxyphenyl)methyl]piperidine-4-carboxylate
4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}-2,1,3-benzoxadiazole
1-{3-[4-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}methyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-2-(1H-indazol-3-yl)-N-(2-methoxyethyl)acetamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-methyl-N-[(3-methyloxetan-3-yl)methyl]-1,2-oxazole-3-carboxamide
5-(azepan-1-yl)-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{[(3-ethoxypropyl)amino]methyl}-4-(6-methoxypyridin-2-yl)phenol
1-{4-[(3-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-phenylethan-1-ol
N-(4-{[1-(3-methoxypropyl)-2,4-dioxo-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}phenyl)acetamide
5-cyclobutyl-N-[(4-methyl-1,4-oxazepan-6-yl)methyl]-1,3,4-oxadiazol-2-amine
3-(1H-indol-3-yl)-N-methyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)propanamide
5-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidine-1-carbonyl)-2,3-dihydro-1H-pyrazol-3-one
2-methoxy-N-[(2R,3R)-2-methoxy-1'-[2-(thiophen-3-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
N-(3-methoxypropyl)-1-methyl-5-[2-(pyridin-4-yl)quinoline-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1,3-dimethyl-N-[3-(pyrrolidin-1-yl)propyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[1-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-2-phenylethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
3-(azocan-1-yl)-N-(2-hydroxy-2-phenylethyl)propanamide
1-(4-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}thiophen-2-yl)ethan-1-one
3-[2-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]propanamide
(1R,3s,6r,8S)-4-[5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-azatricyclo[4.3.1.13,8]undecane
N-[(3R,4S)-4-cyclopropyl-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]-3-(2-oxopiperidin-1-yl)propanamide