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(3S,9aR)-3-(1H-imidazol-4-ylmethyl)-8-(quinolin-5-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(4-hydroxyphenyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1H-pyrazole-5-carboxamide
4-(5-methylpyridin-2-yl)-1-[2-(pyrrolidin-3-yl)benzoyl]piperidin-4-ol
(4-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}morpholin-3-yl)methanol
2,5,6-trimethyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}pyrimidin-4-amine
8-[3-(4-hydroxyphenyl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
6-methyl-4-oxo-N-[3-(pyridin-4-yl)propyl]-4H-pyran-2-carboxamide
N-[(3-methyl-1H-indol-2-yl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[1-(1-cyanocyclopropanecarbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-hydroxy-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(4-methylphenyl)pyrimidine-5-carboxamide
(3S,4S)-1-(3-ethoxypropanoyl)-4-propylpyrrolidine-3-carboxylic acid
2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxamide
8-(5-methyl-1,3,4-thiadiazol-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
8-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{2-[1-(2,7,8-trimethylquinoline-4-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
8-(3,6-dimethylpyrazin-2-yl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidine
2-cyclopropyl-5-[3-(2-methoxyethyl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-3,4-dihydropyrimidin-4-one
N-butyl-N-methyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
1-{2-[2-(2-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}piperidin-2-one
2-{4-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]piperazin-1-yl}-N-phenylacetamide
2-[4-(6-methoxypyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzamido]cycloheptane-1-carboxamide
2-(3-{[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]methyl}phenoxy)ethan-1-ol
N-{[3-methyl-7-(naphthalene-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-sulfonamide
N-({7-[(3-ethoxy-2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
2-[2-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]-1H-imidazole
8-[(3-chloro-5-ethoxy-4-hydroxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
7-cyclohexyl-2-{[6-(dimethylamino)pyridin-3-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-(1-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxy-2-phenylacetamide
N-[2-(dimethylamino)ethyl]-N-(oxolan-2-ylmethyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}thiophene-2-carboxamide
7-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
1-(2-methoxy-4-{[(propan-2-yl)amino]methyl}phenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
ethyl 4-[(3-fluorophenyl)methyl]-1-(oxolane-2-carbonyl)piperidine-4-carboxylate
3-(1-benzyl-1H-imidazol-2-yl)-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidine
2-{1-[(5-methylfuran-2-yl)methyl]-4-(1H-pyrazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
2-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-(5-{[ethyl({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})amino]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
(1S,5R)-N-(3-chloro-4-methoxyphenyl)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-({[(4-fluorophenyl)methyl]amino}methyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)acetamide
N,6-dimethyl-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
1-[1-(methoxymethyl)cyclopropanecarbonyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
N-[(2S,4R,6S)-2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-6-(2-phenylethyl)oxan-4-yl]acetamide
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
(3aR,6aS)-5-(1H-indole-2-carbonyl)-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(5-chloro-2,4-dimethoxyphenyl)methyl](methyl)(oxan-2-ylmethyl)amine