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3-chloro-6-(4-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyridazine
1-(4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
N-methyl-2-[4-(4-methyl-1,4-diazepan-1-yl)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[(5-methylfuran-2-yl)methyl]acetamide
2-[(2-fluorophenyl)methyl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,3-benzoxazole-6-carboxamide
N2-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-N4,N4,5-trimethylpyrimidine-2,4-diamine
(1R,6S)-9-methyl-3-(5-phenyl-1H-pyrrole-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
N-[1-(2,4-dimethylphenyl)propyl]-2-[methyl(piperidin-4-yl)amino]acetamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
1-[(4-chlorophenyl)methyl]-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-6-oxopiperidine-3-carboxamide
3-(4-hydroxyphenyl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
1-(2-chlorophenyl)-5-methyl-4-(5-methylpyrazine-2-carbonyl)piperazin-2-one
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]acetamide
2-[({1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]piperidin-4-yl}oxy)methyl]pyridine
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(1H-indol-3-ylmethyl)methylamine
methyl 3-[3-(5-methylfuran-2-yl)butyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-{[(1,3-dihydroxy-2-methylpropan-2-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
4-(3,3-dimethylpyrrolidine-1-carbonyl)-2-(2-ethylpyrimidin-5-yl)-8-methylquinoline
N-(1-benzyl-2-methyl-7-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-1H-1,3-benzodiazol-5-yl)acetamide
5-[(2,3-difluorophenyl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
1,2,2,6,6-pentamethyl-N-[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperidin-4-amine
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(pyridin-3-yloxy)acetamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-(furan-2-yl)-2-oxoacetamide
[(3-{[1-(2,3-dimethyl-1H-indole-7-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[(4-ethylphenyl)methyl]methylamine
2-methoxy-1-[1'-(pyridin-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
3-(4-methylphenoxymethyl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
5-ethyl-1'-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-methyl-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)butanamide
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-{[2-(trifluoromethyl)phenyl]methyl}propanamide
(1R,3S)-7-(benzenesulfonyl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
1-(3-fluoropyridine-4-carbonyl)-4-(hydroxymethyl)azepan-4-ol
N-[2-(azepan-1-yl)ethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-ethyl-3-{[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]sulfamoyl}-N-(2-methylprop-2-en-1-yl)benzamide
2-acetyl-8-(3-phenylpropanoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
6-{1,9-dioxaspiro[5.5]undecan-4-yl}-2,3-dimethyl-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
3-[1-butyl-3-(carbamoylmethyl)-1H-1,2,4-triazol-5-yl]benzoic acid
4-(2-methoxyphenoxy)-1-(4-methyl-1,3-thiazol-2-yl)piperidine
1-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
5-benzyl-1-(4-methylphenyl)-4-(1,3-thiazole-4-carbonyl)piperazin-2-one
2-(2-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-2-oxoethyl)-5,6-dimethyl-2,3-dihydropyridazin-3-one
5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(pyridin-4-yl)ethyl]-1,2-oxazole-3-carboxamide
3-[(1-benzylpyrrolidin-3-yl)amino]-N-(pyridin-3-yl)propanamide
4-methyl-N-[2-(pyridin-2-ylsulfanyl)ethyl]-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(3-methylbutyl)benzamide
N-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]methyl}-4-(piperidin-1-yl)butanamide
{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(quinolin-2-ylmethyl)amine
3-methyl-7-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one