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2-{3-oxo-9-[(2E)-3-phenylprop-2-en-1-yl]-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
1-[(3-cyanophenyl)methyl]-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
(3S,7S)-5-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
(1S,5R)-6-benzyl-3-(3-fluoro-4-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
7-methoxy-2-[2-(methoxymethyl)pyrimidin-5-yl]-N-(propan-2-yl)quinoline-4-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-2-(dimethyl-1H-1,2,4-triazol-1-yl)acetamide
N-{[4-(methylsulfanyl)phenyl]methyl}-5-propyl-1,3,4-oxadiazol-2-amine
4-[4-(cyclobutylmethyl)piperazine-1-carbonyl]-6-ethyl-2-methylquinoline
[5-({4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)furan-2-yl]methanol
3-[7-(1-hydroxy-2,2-diphenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]pyridin-1-ium-1-olate
{4-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}methanol
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)butanamide
(3S,4R)-4-(3-fluorophenyl)-1-[3-(4-methylpiperazin-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
[(3R,4R)-1-[2-(dimethylamino)-6-(trifluoromethyl)pyrimidin-4-yl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
N,N-diethyl-2-({1-[(4-methoxyphenyl)methyl]-2-oxo-4-(thiolan-3-yl)-1,4-diazepan-6-yl}oxy)acetamide
3-(3-methylphenoxymethyl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
5-[benzyl(methyl)amino]-1-[(4-fluorophenyl)methyl]azepan-2-one
5-{1-[(2-chloro-6-fluorophenyl)methyl]-3-(ethoxymethyl)-1H-1,2,4-triazol-5-yl}-1,2-dihydropyridin-2-one
2-(furan-2-yl)-N-[1-(morpholin-4-ylmethyl)cyclohexyl]-2-oxoacetamide
8-[(2S)-2-amino-2-cyclopropylacetyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-2-yl}-4-methyl-1H-1,3-benzodiazole
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
1-(2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydroquinolin-2-one
4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]-1-[(2E)-2-methylbut-2-en-1-yl]piperidine
(2-{4-[(propan-2-yloxy)methyl]piperidine-1-carbonyl}pyridin-4-yl)methanol
1-(1,4-oxazepan-6-ylmethyl)-3-(2-phenoxyphenyl)urea
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-(1-methyl-1H-pyrazol-4-yl)propanamide
1-(oxan-4-ylmethyl)-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
5-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-2-(propan-2-yl)-1,3-benzoxazole
methyl 1-{9-methoxy-3-[(6-methylpyridin-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperidine-2-carboxylate
(2R,6R)-4-[2-(methylsulfanyl)benzoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-[(2-chloro-6-fluorophenyl)methyl]-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
5-{[2-(4-fluorophenyl)ethyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
methyl 8-(2,1,3-benzothiadiazol-5-ylmethyl)-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
3-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
N-(4-{1-[2-methyl-1-(pyridin-3-yl)propyl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-methyl-1,4-diazepane
1-(5-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
1-(2-methyl-1-benzofuran-5-carbonyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)propane-2-sulfonamide
3-(3-acetylphenyl)-6-[(2-hydroxy-6-methoxyphenyl)methyl]-1-(3-methylbut-2-en-1-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N4,N4,5-trimethyl-N2-[1-(pyridin-3-ylmethyl)piperidin-3-yl]pyrimidine-2,4-diamine
1-(4-benzylpiperidin-1-yl)-3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]propan-1-one
2-(4-fluorophenyl)-N-[3-(methylsulfanyl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
1-methyl-3-[3-(4-{[(1R)-1-phenylethyl]amino}piperidin-1-yl)phenyl]imidazolidin-2-one
N-(2-hydroxy-2-phenylethyl)-1-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
N-[(5-chlorothiophen-2-yl)methyl]-1-(4,7-dimethylquinazolin-2-yl)piperidine-4-carboxamide
7-(2-aminopyridine-4-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-(2-methoxyethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione