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3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[3-(pyridin-3-yl)propyl]propanamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-methyl-2-phenylpropan-1-one
N-(2-methylprop-2-en-1-yl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
5-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1-propylpiperidin-2-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-3-(ethoxymethyl)-1-methyl-1H-1,2,4-triazole
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}({[2-(morpholin-4-yl)pyridin-3-yl]methyl})amine
2-{4-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]piperazin-1-yl}ethan-1-ol
2-chloro-N-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]benzamide
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(1-methoxybutan-2-yl)propanamide
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}urea
5-{3-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-oxopropyl}-5-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidin-2-one
2-(3-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}phenoxy)acetamide
3-[5-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-3-yl)-1,2,4-oxadiazol-3-yl]pyridine
6-(4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazin-1-yl)pyridine-3-carbonitrile
6-methyl-N4-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrimidine-2,4-diamine
8-methoxy-N-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
2-(3-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(4-fluorophenyl)ethyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
4-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-2-(2-methoxyethyl)morpholine
N-[3-(dimethylamino)propyl]-N,2-dimethyl-4-oxo-1,4-dihydroquinoline-8-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
2-[({4-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)amino]-2-methylpropan-1-ol
1-{7-[2-hydroxy-4-(1H-pyrazol-1-yl)butan-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(thiophen-2-yl)ethan-1-one
2-[methyl(pyridin-3-ylmethyl)amino]-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
2-(4-chlorophenyl)-4-(2-propyl-1,3-thiazole-4-carbonyl)morpholine
1-(3-methylpyrazin-2-yl)-4-(pyridin-3-yl)piperidin-4-ol
methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl][(3-{[1-(thiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]amine
2-{4-[1-(2-hydroxyethyl)piperidine-3-carbonyl]piperazin-1-yl}benzonitrile
1-methyl-4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
5-[(3-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2-oxazole-3-carboxamide
(1S,5R)-6-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carboxamide
(3S,4R)-3-methoxy-1-{[1-phenyl-3-(pyridin-4-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-amine
(2S,4S)-N-ethyl-1-(oxan-4-yl)-4-[(2E)-3-phenylprop-2-enamido]pyrrolidine-2-carboxamide
N-cyclopentyl-3-{[(5-methyl-1,2-oxazol-3-yl)methyl]sulfamoyl}benzamide
[(3R,4R)-1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
2-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-N-(2-phenylethyl)acetamide
methyl (1R,3S,3aR,6aS)-1-ethyl-5-methyl-3-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
9-ethyl-4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl 2-(4-{5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carbonyl}morpholin-3-yl)acetate
2-(4-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol
1-{3-[1-(dimethylamino)ethyl]phenyl}naphthalen-2-ol
2-cyclopentyl-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}acetamide
(2S,4R)-4-amino-N-methyl-1-[(1-propyl-1H-imidazol-2-yl)methyl]pyrrolidine-2-carboxamide
2-{3-[2-(methylsulfanyl)ethyl]-5-[1-(2-oxopyrrolidin-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
N-ethyl-1-{[5-(methoxymethyl)furan-2-yl]methyl}-N-(pyridin-4-ylmethyl)piperidin-3-amine
(2S)-1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-2-phenylethan-1-one
3-({2-[1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}(methyl)amino)-1λ6-thiolane-1,1-dione
3-{[(3-methylpyridin-2-yl)methyl]sulfamoyl}-N-[(2R)-pyrrolidin-2-ylmethyl]benzamide
3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidine