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N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,3,3-trifluoropropanamide
(1S,6R)-9-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
5-({ethyl[(4-ethylphenyl)methyl]amino}methyl)-2-methoxyphenol
1-methyl-9-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-1,4,9-triazaspiro[5.5]undecan-5-one
4-pentyl-3-(1H-pyrazol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(3-methoxyphenyl)phenyl]-1-(3-methylpyrazin-2-yl)piperidine-4-carboxamide
1-{3-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-propoxyethan-1-one
N-[(2,3-dimethoxyphenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
3-[1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-yl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{1-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
1-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
2-[2-({[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}amino)ethyl]-3,4-dihydroquinazolin-4-one
2-cyclohexyl-5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)pyrimidine
4-methyl-3-oxo-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
(2R,4S)-1-(3-chloro-5-methoxybenzoyl)-4-hydroxypiperidine-2-carboxylic acid
4-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
9-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 2-(4-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)acetate
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-(1H-pyrazol-1-yl)propanamide
9-[(2-aminopyridin-3-yl)methyl]-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
8-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(4-sulfamoylphenyl)methyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-3-(4H-1,2,4-triazol-4-yl)propanamide
3-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-imidazol-2-yl}-2-(morpholin-4-yl)quinoline
1-cyclohexyl-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}piperidine-3-carboxamide
1-[(2,6-dimethoxyphenyl)methyl]-4-(1-ethyl-1H-pyrazol-4-yl)-1H-1,2,3-triazole
N,N-diethyl-1-{1-[4-(furan-2-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}pyrrolidin-3-amine
2-(9-{[4-(3-hydroxyprop-1-yn-1-yl)phenyl]methyl}-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl)acetamide
N-cyclopropyl-3-[5-(2-phenoxyacetyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
7-(1,3-benzothiazol-2-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-4-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]-1,4-diazepan-2-one
3-{1-[(2,4-difluorophenyl)methyl]piperidin-3-yl}-N-[(2,4-dimethoxyphenyl)methyl]propanamide
N-(5-fluoropyridin-3-yl)-2-methyl-4-[(3-methylphenyl)methyl]-3-oxopiperazine-1-carboxamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
1-methyl-5-{[2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}piperidin-2-one
N-benzyl-N-(cyclopropylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetamide
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amine
N-[4-(morpholin-4-ylmethyl)phenyl]-4-(4H-1,2,4-triazol-3-yl)piperidine-1-carboxamide
2-(1-methyl-6-oxo-1,6-dihydropyridine-3-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-{2-[1-ethyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylbenzene-1-sulfonamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{2-[4-(propan-2-yloxy)phenyl]ethyl}acetamide
8-(1H-indol-2-ylmethyl)-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine-4-carboxamide
N-[1-(4-{[2-(cyclohex-1-en-1-yl)ethyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]oxolane-3-carboxamide
4,4-difluoro-N-[3-(1H-imidazol-5-yl)phenyl]piperidine-1-carboxamide
4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidine