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N-[(5-chlorothiophen-2-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[(1-methylpiperidin-4-yl)methyl]-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperazine
N3-(adamantan-1-ylmethyl)-1-benzyl-N5-cyclopropyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[5-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
5-benzyl-1-(4-methylphenyl)-4-(2-oxo-2,3-dihydro-1H-imidazole-4-carbonyl)piperazin-2-one
[(3R,4S)-4-(morpholin-4-ylmethyl)-1-[(4-phenylphenyl)methyl]pyrrolidin-3-yl]methanol
6-cycloheptyl-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N-[(2R)-1-{4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-1-oxopropan-2-yl]acetamide
1-[2-(1H-imidazol-4-yl)ethyl]-5-(oxan-4-yl)-4-phenyl-1H-imidazole
7-(3-chlorophenyl)-4-cyclopropanecarbonyl-9-(thiophen-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
[(1-cyclopentylpiperidin-4-yl)methyl]({[4-(methylsulfanyl)phenyl]methyl})(pyridin-3-ylmethyl)amine
2-{3-[({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]phenyl}ethan-1-amine
1-[(5-methylfuran-2-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
N-(1-{1-[(2R)-2-amino-4-methylpentanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
2-(1-benzyl-1H-pyrazol-4-yl)-2-(4-cyclopentyl-3-oxopiperazin-1-yl)acetic acid
1-{2-methyl-2,8-diazaspiro[4.5]decan-8-yl}-2-(piperazin-1-yl)ethan-1-one
2-(4-{[methyl({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}piperidin-1-yl)ethan-1-ol
(1s,4s)-N-[(3,5-dimethoxyphenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]cyclohexan-1-amine
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetamide
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pent-2-yn-1-yl)pyrrolidin-3-yl]-1-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
(3S,4R)-1-[2-(dimethylamino)benzoyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
9-[2-(1,4-dimethylpiperazin-2-yl)acetyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
1-(3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzoyl)azetidin-3-ol
[(4-chlorophenyl)methyl]({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
1-cyclohexyl-4-(3-methylbut-2-enoyl)piperazin-2-one
4-{[2-(ethylamino)pyrimidin-5-yl]methyl}-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(6-methoxynaphthalen-2-yl)-4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}morpholine
3-{2-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
2-{4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]butyl}pyridine
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}(2,1,3-benzothiadiazol-5-ylmethyl)methylamine
2-(pyridin-3-yl)-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]pyrimidine
1-[2-(4-methoxyphenyl)ethyl]-N,N-dimethyl-5-(1H-pyrazol-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{4-[5-fluoro-4-(methylamino)pyrimidin-2-yl]phenyl}methanol
3-(ethylsulfanyl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(4-methylpyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(4-methoxyphenyl)-5-[4-(methylsulfanyl)butan-2-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
4-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3R,4R)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
4-{[5-(1-benzoylpiperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
4-[3-(4-methylpiperidine-1-carbonyl)piperidin-1-yl]-2-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
[5-({1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl}methyl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(6-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[2-(dimethylamino)-6-(2-methylphenyl)pyridine-3-carbonyl]piperazine-1-carbaldehyde
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1H-imidazol-2-yl)-1H-1,2,3-triazole
6-methyl-5-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}quinoline
1-{3-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
N,2,4,5-tetramethyl-N-[2-(2-oxopiperidin-1-yl)ethyl]benzamide
2-fluoro-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-5-sulfamoylbenzamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(1H-pyrazol-1-yl)benzamide