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1-butyl-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazin-2-one
N-[(1R,3S)-3-(pyrrolidine-1-carbonyl)cyclopentyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
7-fluoro-3-({[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}methyl)-1,2-dihydroquinolin-2-one
1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-4-phenoxypiperidine-4-carboxylic acid
3-amino-1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
ethyl 1-[2-(furan-2-yl)-2-oxoacetyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
5-ethyl-6-methyl-N4-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyrimidine-2,4-diamine
3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-methylurea
N-(5-{[(cyclobutylmethyl)(oxolan-2-ylmethyl)carbamoyl]amino}-2-methoxyphenyl)acetamide
7-(furan-2-ylmethyl)-N-(1H-imidazol-2-ylmethyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
ethyl 4-[1-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
2-(3,4-dichlorophenyl)-N,N-diethylmorpholine-4-carboxamide
3-methyl-1-(2-methylpropyl)-4-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]piperazin-2-one
methyl 2-[2-(2-{[1-(furan-2-yl)ethyl]amino}acetamido)-1,3-thiazol-5-yl]acetate
(1,4-dioxan-2-ylmethyl)[(3-fluoro-4-methoxyphenyl)methyl]methylamine
ethyl 1-[(2S)-1-acetylpyrrolidine-2-carbonyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
1-(2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}pyrimidin-4-yl)piperidin-4-ol
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-(3,4-dihydro-2H-1-benzopyran-3-yl)acetamide
(1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-4-yl)(pyridin-2-yl)methanol
N-methyl-N-(1-methylpiperidin-4-yl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
ethyl 5-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-(2,2,2-trifluoroethyl)piperidine-3-carboxamide
1-phenyl-N,N-bis(pyridin-3-ylmethyl)-1H-1,2,3-triazole-5-carboxamide
(2S,4R)-4-amino-N-methyl-1-[(3-methylthiophen-2-yl)sulfonyl]pyrrolidine-2-carboxamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-(dimethylamino)butan-1-one
1-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-3-(2-methoxyphenyl)propan-1-one
2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-(9H-fluoren-9-yl)acetamide
(1S,5R)-6-methyl-3-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
(3R,4R)-1-[(2-methyl-1H-imidazol-4-yl)methyl]-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
N-{1-[1-(3,3-dimethylbutanoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
1-({2,5-dimethyl-3-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)-N-methylpyrrolidine-3-carboxamide
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-5-(4-methylphenyl)-1H-pyrazole-3-carboxamide
1-(oxan-4-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-3-carboxamide
[(3R,4S)-1-[(3-fluorophenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
(2S,4S)-4-amino-1-methyl-N-[3-(morpholin-4-yl)propyl]pyrrolidine-2-carboxamide
2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]acetamide
2-methyl-5-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]pyrazine
1-[3-(5-methylfuran-2-yl)benzoyl]-4-(pyridin-3-ylmethyl)piperazine
1-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-6-oxo-N-(oxolan-2-ylmethyl)-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-methyl-6-[3-methyl-5-(2-propyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-1-yl]pyridine
[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
4-{4-[(2,4-dimethylphenyl)methyl]piperazin-1-yl}-5-ethyl-2-methylpyrimidine
5-(cycloheptylamino)-N,N-dimethyl-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[9-(6-methylpyridine-3-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
2-methyl-1-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)azetidin-3-yl]piperidine
[1-(2,5-dimethylfuran-3-carbonyl)-3-[(4-fluorophenyl)methyl]piperidin-3-yl]methanol
1-[6-(1H-indol-5-yl)pyridin-3-yl]ethan-1-one
6-(3-aminopyrrolidin-1-yl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzamide