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2-chloro-5-(1H-pyrazol-1-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
3-(benzenesulfonyl)-1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]propan-1-one
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
1-[5-(2-benzylmorpholine-4-carbonyl)thiophen-2-yl]ethan-1-one
5-[2-(aminomethyl)-5-chloro-2,3-dihydro-1-benzofuran-7-yl]thiophene-2-sulfonamide
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
N-[cyclopropyl(4-methoxyphenyl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-({2-[(5-ethyl-2-methylpyrimidin-4-yl)amino]ethyl}amino)-6-methyl-3,4-dihydropyrimidin-4-one
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
2-({4-[4-(pyridin-4-yl)piperidine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
2,6-dimethyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]quinoline-3-carboxamide
1-methyl-3-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-5-(thiophen-2-yl)-1H-pyrazole
1,6-dimethyl-N-{2-[methyl(2-phenylethyl)amino]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(2-ethylbutyl)-8-(1-ethylpyrrolidine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{5-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl}acetic acid
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-(4-fluoro-2-methylphenyl)propanamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[3-(methylsulfanyl)propyl]acetamide
2-[(2-ethylpiperidin-1-yl)methyl]-4-(pyridin-2-yl)phenol
1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
1-(dimethylamino)-3-(4-methoxy-2-{6-oxa-9-azaspiro[4.5]decan-9-ylmethyl}phenoxy)propan-2-ol
N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]furan-3-carboxamide
5-{1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
N-{3-[2-(dimethylamino)acetamido]-4-methylphenyl}azocane-1-carboxamide
(2S,4R)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-1-[(4-ethylphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(2-ethoxyethyl)-1-[(2-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
(2E)-1-[3-(5-benzyl-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(4-methoxyphenyl)prop-2-en-1-one
3-methyl-1-{4-[methyl(oxan-2-ylmethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}but-2-en-1-one
1-methyl-3-[1-(1-methylpiperidin-4-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]piperidine
N-(butan-2-yl)-N-[(2-chlorophenyl)methyl]-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
2-(1-butyl-3-methyl-1H-1,2,4-triazol-5-yl)-5-methyl-1H-indole
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
5-ethyl-4-methyl-6-{4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}pyrimidin-2-amine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4,6-dimethyl-1-(2-{[1-(2-methylphenyl)piperidin-4-yl]amino}ethyl)-1,2-dihydropyrimidin-2-one
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)furan-2-carboxamide
1,3-dimethyl-5-(1-phenyl-1H-pyrazol-4-yl)-1H-1,2,4-triazole
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-2-ylmethyl)benzamide
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-5,6,7,8-tetrahydroquinoline-3-carboxamide
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
1-[1'-(1-ethyl-1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[3-(2-methoxyphenyl)-1H-pyrazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
5-chloro-3-phenyl-2-(thiomorpholine-4-carbonyl)-1H-indole
N-(6-aminohexyl)-2-methyl-1-benzofuran-5-carboxamide
1-(4-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}thiophen-2-yl)ethan-1-one
3-(morpholine-4-carbonyl)-N-[(1-phenylcyclohexyl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(azocan-1-yl)-3-(4-{[4-(2-hydroxyethyl)piperidin-1-yl]methyl}-2-methoxyphenoxy)propan-2-ol
2-(dimethylamino)-2-(2-fluorophenyl)-N-[3-(4-methylpiperazin-1-yl)propyl]acetamide