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N-{3-[2-(4,5-dimethylfuran-2-yl)-1H-imidazol-1-yl]-2-methylphenyl}-2-methoxyacetamide
3-{[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyridine
methyl 3-{[(3-ethyl-1-methyl-1H-pyrazol-5-yl)formamido]methyl}-5-[3-(trifluoromethyl)benzamido]benzoate
(1S,5R)-3-(3-propyl-1H-pyrazole-4-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-cyclohexyl-1,4-diazepan-1-yl)-2-[4-(3-hydroxypropyl)phenyl]acetic acid
1-[1-(1-ethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]-1H-pyrazole-4-carboxamide
N,4-dimethyl-5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1,3-thiazol-2-amine
1-(2-chloro-4,6-dimethylphenyl)-3-[3-(oxolan-3-yl)propyl]urea
methyl (2S,3S)-2-({5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazol-3-yl}formamido)-3-methylpentanoate
3-[3-(2-phenylacetyl)piperidine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
(1S,4S)-5-(3-fluorobenzoyl)-2-(2-methyl-1,3-benzothiazol-5-yl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-methoxy-N-[(2R,3R)-1'-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
1-cyclobutanecarbonyl-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
(2S,4S)-4-amino-1-(azepane-1-sulfonyl)-N,N-diethylpyrrolidine-2-carboxamide
2-(1H-indol-1-yl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]ethan-1-one
N-cyclohexyl-2-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}quinazolin-4-amine
4-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]pyrrolidin-3-yl}-2-(pyridin-4-yl)pyridine
1-[benzyl(methyl)amino]-3-[4-({[2-(piperidin-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
methyl 1-ethoxy-2-oxo-8-(4-oxo-4-phenylbutanoyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
6-methyl-N-(2-methylpropyl)-2-oxo-N-(3-phenylprop-2-yn-1-yl)-1,2-dihydroquinoline-4-carboxamide
2-[3-(2,4-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-3-methylpyridine
N-(4-methoxyphenyl)-1-{2-[2-(3-methoxyphenyl)acetamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
(3S)-4-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-ethyl-3-methylpiperazin-2-one
(3R,4R)-4-amino-1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-3-ol
N-(2,4-dimethoxyphenyl)-2-(4-methyl-1,4-diazepan-1-yl)pyridine-3-carboxamide
2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]-N-(3-phenylpropyl)acetamide
2-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)ethan-1-ol
(2S,4S)-4-amino-1-[(2R)-oxolane-2-carbonyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(1S,5R)-6-(3-fluorobenzoyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-methoxy-6-(2-methylpyrimidin-4-yl)-N,N-bis(propan-2-yl)benzamide
1-cyclopentyl-4-oxo-N3-(prop-2-en-1-yl)-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
4-({[2-(dimethylamino)-1-phenylethyl](methyl)carbamoyl}amino)-N,N,3-trimethylbenzamide
(3S)-3-benzyl-4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
2-(2-{[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrrol-1-yl)pyridine
3-methyl-6-[4-(piperidin-1-ylmethyl)piperidin-1-yl]pyridazine
1-{3-[2-({[(5-fluoro-2-methylphenyl)methyl]amino}methyl)-4-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
ethyl 4-[(2-chlorophenyl)methyl]-1-[(2-hydroxyphenyl)methyl]piperidine-4-carboxylate
methyl 9-(2,3-dihydro-1H-inden-2-yloxy)-3-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(3-hydroxy-2,2-dimethylpropyl)piperidine-3-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}propanamide
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(pyridin-3-yloxy)ethan-1-one
N-benzyl-5-({[2-(1H-imidazol-1-yl)ethyl](methyl)amino}methyl)pyrimidin-2-amine
7-[(3-methylphenyl)methyl]-2-(1-methylpiperidin-4-yl)-2,7-diazaspiro[4.5]decane
N4-[(1-benzylpyrrolidin-3-yl)methyl]-N4,6-dimethyl-5-(prop-2-en-1-yl)pyrimidine-2,4-diamine
N-[2-(dimethylamino)ethyl]-5-(4-methylpyridine-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
methyl (2S)-1-[2-cyclobutyl-5-(2-methoxyacetamido)-1-methyl-1H-1,3-benzodiazole-7-carbonyl]pyrrolidine-2-carboxylate
4-{4-[(2,3-dimethyl-1H-indol-7-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
3-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl](methyl)amino}propane-1,2-diol