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N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methylacetamide
1-cyclopentyl-N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxamide
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-(pyridin-2-ylmethyl)piperazine
N4-[(2-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
1-[(3-chlorophenyl)methyl]-5-(2,2-dimethyloxan-4-yl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(3,4-dimethoxyphenyl)methyl]amine
2-hydroxy-N-methyl-4-(methylsulfanyl)-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}butanamide
N-cyclohexyl-4-(piperidin-3-yl)-N-(pyridin-2-ylmethyl)benzamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-4-(1H-pyrazol-4-yl)butanamide
2-benzyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1,3-thiazole-4-carboxamide
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[2-(propan-2-yl)pyrimidin-5-yl]methyl}amine
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,3-oxazole
1-(3-cyano-4-methoxyphenyl)-3-ethyl-3-(2,2,2-trifluoroethyl)urea
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
1-[5-({1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}carbonyl)thiophen-2-yl]ethan-1-one
3-(4H-1,2,4-triazol-4-ylmethyl)quinoline
N,4-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]piperazine-2-carboxamide
2-(4-{[2-(dimethylamino)ethyl](methyl)amino}piperidin-1-yl)-2-(2,4-dimethylphenyl)acetic acid
5-amino-N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-4-phenyl-1H-pyrazole-3-carboxamide
methyl 4-({1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidin-3-yl}formamido)butanoate
(3aS,6aS)-2-acetyl-5-(5-propyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-cyclopropyl-2-(pyrrolidin-1-yl)-6-(trifluoromethyl)pyrimidin-4-amine
4-chloro-N,2,5-trimethyl-N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}benzene-1-sulfonamide
4-({3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-6,7-dimethyl-2H-chromen-2-one
6-(2-chloro-4-fluorophenyl)-4-(4-methylpiperazin-1-yl)quinazoline
1-[6-(2-methylphenyl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
1-(2-methylfuran-3-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
2-(4-{2-[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]-1H-imidazol-1-yl}piperidin-1-yl)pyridine-3-carbonitrile
5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-imidazole
N,1-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrrole-2-carboxamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}acetic acid
5-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
methyl 2-{8-[(4-acetamidophenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
1-cyclohexyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-(3-chlorophenyl)urea
(4aS,8aR)-6-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
4-(4-methoxypyrimidin-2-yl)-N-(1-methyl-1H-indazol-6-yl)piperazine-1-carboxamide
2-{2-[1-(2-hydroxynaphthalene-1-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
1-(4-oxo-4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}butyl)piperidin-2-one
N-[1-(1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
(4aS,7aR)-1-benzoyl-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-cyclohexyl-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-1H-pyrazole-4-carboxamide
methyl 3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-5-[(pentan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(3-fluorophenoxymethyl)-N-methyl-N-(1H-pyrazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
(4aS,8aS)-2-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-decahydroisoquinolin-4a-ol
6,7-dimethoxy-1-[(4-methylphenyl)methyl]-3-({[3-(2-oxopyrrolidin-1-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
3-(4-methoxyphenyl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1H-pyrazole-5-carboxamide
2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]acetamide
2-(3-methylbut-2-en-1-yl)-8-[3-(pyridin-3-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one