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N-[(3-chlorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
1-[4-(2-methylphenyl)piperazin-1-yl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(pyridin-2-ylmethyl)piperidin-3-yl]propan-1-one
(1R,3S)-7-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-7-azaspiro[3.5]nonane-1,3-diol
(2S)-2-[2-(2,3-dichloro-4-methylphenyl)-1H-imidazol-1-yl]-3-methylbutanamide
5-(2,6-dimethylphenoxymethyl)-N-(oxolan-3-yl)-1,2-oxazole-3-carboxamide
2-[(4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]phenol
2-[(cyclopropylmethyl)sulfanyl]-1-[4-(4-methoxybenzoyl)piperazin-1-yl]ethan-1-one
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-methylpyrimidine-5-carboxamide
1-[1-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)pyrrolidin-3-yl]-3,5-dimethyl-1H-pyrazole
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}benzenesulfonamide
N-[3-(2-chlorophenoxy)propyl]-N,2-dimethyl-1,3-benzoxazole-6-carboxamide
dimethyl({[(3S,4R)-1-[2-(methylsulfanyl)pyrimidin-4-yl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
1-(4-{[4-(5-methyl-1H-indole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazin-1-yl)ethan-1-one
(2E)-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enamide
N-[(3S,4R)-4-propyl-1-(9H-purin-6-yl)pyrrolidin-3-yl]methanesulfonamide
1-[(4-{[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]-4-phenylpiperidine
1-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyridin-4-yl)piperazine
1-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)urea
N-[2-(1-ethylpiperidin-4-yl)ethyl]-3-(3-hydroxy-3-methylbutyl)benzamide
9-(6,8-dimethylquinolin-4-yl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
2-amino-1-[2-(4-chlorophenyl)morpholin-4-yl]ethan-1-one
1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
3-(1-ethyl-1H-imidazol-2-yl)-1-[4-(5-methylfuran-2-yl)benzoyl]piperidine
4-({ethyl[(3S,4R)-4-hydroxyoxolan-3-yl]amino}methyl)-N-(6-methylpyridazin-3-yl)benzamide
2-({[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[1-(thiophen-3-yl)propan-2-yl]piperidine-4-carboxamide
methyl[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-(naphthalen-1-yl)-5-(oxolan-2-ylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-[(5-phenylthiophen-2-yl)methyl]pyrrolidin-3-yl]methanol
2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
4-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}thiomorpholine
5-({3-[4-(pyridin-2-ylmethyl)piperazine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)isoquinoline
N-{1-[1-(adamantane-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[3-(3-methylphenyl)phenyl]piperidin-4-amine
N-{[2-(2-benzamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
methyl[(2-methyl-1H-imidazol-4-yl)methyl]{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
4-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-2-methyl-1,4-oxazepane
4-cyclopentyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]pyrimidin-2-amine
methyl 3-[(3,4-dimethylphenyl)methyl]-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-(4-{[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-1H-indole
4-methanesulfonyl-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)benzamide
3-{[1-(2-methanesulfonamidoacetyl)pyrrolidin-3-yl]methyl}benzamide
3-{[1-(2-aminopyridine-4-carbonyl)piperidin-4-yl]methyl}benzoic acid
3-[1-(6-aminopyrimidin-4-yl)piperidin-4-yl]-4-benzyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(2,2-diphenylethyl)-2-(methylamino)pyridine-4-carboxamide
methyl 4-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]carbamoyl}butanoate
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-8-methyl-1,4-dihydroquinolin-4-one
4-[4-(2,4-dimethylphenyl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one