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(furan-2-ylmethyl)({[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl})(prop-2-yn-1-yl)amine
methyl 2-(5-methyl-2-{[(4-methyl-1,2,3-thiadiazol-5-yl)formamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
methyl (2S,4S)-1-[(2-ethoxyphenyl)methyl]-4-(2-fluorobenzamido)pyrrolidine-2-carboxylate
2-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]pyridine-3-carboxylic acid
6-chloro-N,N-dimethyl-3-{[methyl(1-methylpyrrolidin-3-yl)amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl](methyl)[3-(pyrrolidin-1-yl)butyl]amine
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-N'-(2,5-dimethylphenyl)propanediamide
(1S,5R)-3-methyl-6-[(5-propylfuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}acetamide
4-[5-(morpholin-2-ylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]benzamide
N-[(4-sulfamoylphenyl)methyl]-2-(4H-1,2,4-triazol-4-yl)benzamide
2-(adamantan-1-yl)-5-[4-(aminomethyl)piperidine-1-carbonyl]pyrimidin-4-ol
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[2-(4-methylphenoxy)ethyl]propanamide
1-[4-({[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]amino}methyl)piperidin-1-yl]ethan-1-one
3-[4-({2-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)piperazin-1-yl]propanamide
4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-N-(thiophen-3-ylmethyl)pyrimidin-2-amine
4-{5-methanesulfonyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-5-methyl-3-phenyl-1,2-oxazole
2-{5-[(2,2-dimethyloxan-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-1,3-benzodiazole
5-ethyl-2-{1-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}pyridine
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1H-imidazole-2-carboxamide
4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}-6-methyl-2-propylpyrimidine
1-cyclopentyl-N-(diphenylmethyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-ethyl-4-{[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyrimidine
N-cyclopentyl-3-[5-(cyclopentylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
2-(2H-1,3-benzodioxol-5-yl)-4-[1-(furan-2-ylmethyl)pyrrolidin-3-yl]pyridine
(3S,4R)-1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-[1-(2,2-dimethylpropyl)-4-(1H-indol-2-ylmethyl)piperazin-2-yl]ethan-1-ol
5-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]quinoxaline
2-methyl-4-(5-{[methyl({[1-(2-methylpropyl)piperidin-4-yl]methyl})amino]methyl}thiophen-2-yl)but-3-yn-2-ol
N-(2-methylprop-2-en-1-yl)-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
6-(2-fluoro-4-methoxyphenyl)-N-[(2S)-1-hydroxypropan-2-yl]-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-[(3S)-3-hydroxy-3-phenylpropyl]-1-(4-methoxyphenyl)piperazin-2-one
({4-[(1-cyclohexanecarbonylpiperidin-4-yl)oxy]phenyl}methyl)(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
1-(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carbonyl)azocane
4-(4-methoxyphenyl)-3-[3-(morpholin-4-yl)propyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4S)-1-(oxane-4-carbonyl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
3-[3-(3-methoxyphenoxy)azetidin-1-yl]-6-phenylpyridazine
N-(2-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}ethyl)pyridine-3-carboxamide
1-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)ethan-1-one
4-(2-phenoxyethyl)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1,4-diazepan-5-one
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(1-methyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2-fluorophenyl)-3-phenyl-1-[4-(pyridin-4-yl)piperazin-1-yl]propan-1-one
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
4-fluoro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)benzamide
5-(2-methylpropyl)-5-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
1-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)pyrrolidin-2-one
3-[3-(1-ethyl-1H-pyrazol-4-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
N-{[7-(1H-indol-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}oxolane-3-carboxamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide