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(1r,4r)-N-({1-[(2-ethylpyrimidin-4-yl)methyl]pyrrolidin-3-yl}methyl)-4-methylcyclohexane-1-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(quinoline-6-carbonyl)-decahydro-1,6-naphthyridin-2-one
(1R,3S)-3-{4-[(pyridin-2-ylmethyl)carbamoyl]piperidine-1-carbonyl}cyclopentane-1-carboxylic acid
4-[(3-ethoxy-4-methoxyphenyl)methyl]-8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-4-(pyrazin-2-yl)-1,4-diazepan-6-ol
N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]cyclopropanecarboxamide
6-[2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]-N-(propan-2-yl)pyrimidin-4-amine
1-[1-(1-phenylmethanesulfonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
(2S)-2-(2,3-difluorophenyl)-2-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}acetic acid
1-[3-(4-tert-butylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
N-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-{4-[4-phenyl-1-(pyridin-3-ylmethyl)-1H-imidazol-5-yl]phenyl}acetamide
1-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-2-(2-methoxyphenoxy)ethan-1-one
N-cyclopropyl-5-[2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
5-methoxy-2-{[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}pyridin-4-ol
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(3-fluoro-4-methoxyphenyl)-1H-indazol-1-yl]acetamide
5-chloro-N-(3-methyl-4-pentanamidophenyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
[(3R,4R)-4-(morpholin-4-ylmethyl)-1-(3-propyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methanol
4-{[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
methyl 2-[8-(2,2-dimethylpropyl)-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)propanamide
N-(2H-1,3-benzodioxol-5-yl)-2-{4-[(5-propylfuran-2-yl)methyl]morpholin-3-yl}acetamide
4-(2,3-dihydro-1-benzofuran-2-carbonyl)-7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3,5-dimethyl-1-[(4-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)methyl]-1H-pyrazole
(2S)-2-{[4-({[1-(hydroxymethyl)cyclopropyl]methyl}(methyl)sulfamoyl)phenyl]formamido}propanamide
ethyl 5-(2,4-dimethoxyphenyl)pyridine-3-carboxylate
1-(3,5-dichloro-4-methylbenzoyl)-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]cyclobutanecarboxamide
ethyl 3-{[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]amino}-6-methylthieno[2,3-b]pyridine-2-carboxylate
methyl 4-[4-({[1-(4-methoxyphenyl)ethyl](methyl)amino}methyl)-5-methyl-1,3-oxazol-2-yl]benzoate
3-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]naphthalen-2-ol
4-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]oxane-4-carbonitrile
N-(1,4-dioxan-2-ylmethyl)-2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
N-methyl-N-(thiophen-3-ylmethyl)-1H-1,2,3-benzotriazole-5-carboxamide
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)-1-(4,4,4-trifluorobutyl)piperidine
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-(piperidin-1-yl)butanamide
4-(1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-yl)benzoic acid
2-({4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepan-1-yl}methyl)benzoic acid
1-[(4aR,8aS)-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-(4-methoxyphenyl)ethan-1-one
4-[5-(methoxymethyl)furan-2-carbonyl]-7-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 1-[2-(2-oxopiperidin-1-yl)acetyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
N2,N2,N4,5,6-pentamethyl-N4-(oxolan-2-ylmethyl)pyrimidine-2,4-diamine
1,1,1-trifluoro-3-{3-[3-(3-methylpyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}propan-2-ol
2-ethyl-N-{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}-4-methyl-1,3-oxazole-5-carboxamide
3-hydroxy-3-({[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide