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2-(trimethylpyrimidin-4-yl)benzamide
N-{3-[3,5-dimethyl-1-(2-oxopropyl)-1H-pyrazol-4-yl]phenyl}acetamide
1-{4-[7-(5,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidin-1-yl}ethan-1-one
(1R,5R)-3-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonane
methyl 7-oxo-9-(propan-2-yloxy)-3-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-(3-fluorophenyl)-N-{[4-methoxy-3-(pyridin-3-ylmethoxy)phenyl]methyl}-N-[(3S)-2-oxoazepan-3-yl]benzamide
[2-(2-phenylphenyl)-1,3-thiazol-4-yl]methanol
(2S)-N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)pyrrolidine-2-carboxamide
6-methyl-5-[3-(2-methylphenyl)piperidine-1-carbonyl]-2-oxo-1,2-dihydropyridine-3-carbonitrile
4-[(4-ethoxyphenyl)methyl]-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]piperazin-2-one
5-(2-ethylpyrimidine-5-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-({7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
4-benzoyl-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidine
methyl (2S,4R)-1-benzyl-4-(2,3-dimethyl-1H-indole-7-amido)pyrrolidine-2-carboxylate
2-acetyl-8-(1,3-thiazol-4-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
8-fluoro-2-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}quinolin-4-ol
6-(2-chlorophenyl)-7-(cyclopropylmethyl)-N-(2,2-difluoroethyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-cyclohexyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1H-pyrazole-4-carboxamide
5-(2-chlorophenyl)furan-2-carboxamide
[2-(1H-indol-4-yl)quinolin-3-yl]methanol
3-({4-[3-(3,3-diethylpyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-(4-chlorophenyl)-4-[(2-propylpyrimidin-5-yl)methyl]morpholine
(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl){[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
2-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
1-(cyclopropylmethyl)-3-(2,3-dimethoxyphenyl)-6-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
3-({[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)pyrrolidin-3-ol
4-hydroxy-2-({methyl[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)quinoline-6-carboxamide
1-(5-acetyl-2-ethoxyphenyl)-3-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)urea
4-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
9-methanesulfonyl-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(azetidine-1-carbonyl)benzenesulfonyl]-3-(methoxymethyl)pyrrolidine
[(3R,4S)-1-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
1-[(1S,5R)-6-(2-chlorobenzoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-(1-methylpiperidin-2-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
2-{4-[(2-butyl-1H-imidazol-4-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
4-[4-(1H-indol-5-ylmethyl)-2-oxopiperazin-1-yl]benzonitrile
(2S,4S)-4-amino-1-({1-[(2-chlorophenyl)methyl]-1H-1,3-benzodiazol-2-yl}methyl)pyrrolidine-2-carboxylic acid
1-(2,6-dimethoxypyridine-3-carbonyl)-3-[(dimethylamino)methyl]piperidin-3-ol
2-(4-chloro-2-methylphenoxy)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
1-(2,3-dihydro-1H-indene-1-carbonyl)-4-(3-methoxybenzoyl)piperazine
1-(5-phenyl-1,3,4-thiadiazol-2-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]piperidin-4-amine
5-(2-fluoro-6-methoxyphenyl)-3-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
2-[1-(2-methoxyphenyl)-5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepin-9-yl}-1H-1,2,4-triazol-3-yl]acetamide
(4aS,7aR)-1-benzoyl-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}({1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
8-cyclopropanecarbonyl-2-(3-methoxybenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-methoxy-N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)benzamide