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[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(3-methylpyridin-4-yl)pyrrolidin-3-yl]methanol
3-(3-{1-[(3,5-dimethylphenyl)formamido]-3-methylbutyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl)pyridin-1-ium-1-olate
1-(3,5-dimethylbenzoyl)-4-ethyl-1,4-diazepan-5-one
7-(4-chloro-1H-pyrazole-3-carbonyl)-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(carbamoylamino)-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]acetamide
N-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
1-(cyclohexylmethyl)-5-(3-methylpiperidin-1-yl)azepan-2-one
2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(2-methylpropyl)acetamide
(4aS,8aR)-1-(3-hydroxypropyl)-N-[(3-methylphenyl)methyl]-2-oxo-decahydro-1,6-naphthyridine-6-carboxamide
4-(azocane-1-carbonyl)-6-fluoro-2-(2-methylpyrimidin-5-yl)quinoline
4-[(4aR,8aR)-6-(3-phenylpropanoyl)-decahydro-1,6-naphthyridine-1-carbonyl]-2-methyl-1,2-dihydrophthalazin-1-one
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-6-methylpyridine-2-carboxamide
1-[(4-chlorophenyl)methyl]-N-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-({7-[2-(cyclohex-1-en-1-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(phenylsulfanyl)acetamide
(1R,5R)-6-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[1-(thiophen-2-yl)ethyl]piperidine-4-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-1-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}ethan-1-one
N-({8-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
N-(2,4-difluorophenyl)-3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidine-1-carboxamide
4-(4-acetyl-3-fluorophenoxy)-1-cycloheptylpiperidine-4-carboxylic acid
7-fluoro-2-methyl-4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]quinoline
3-benzyl-4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}benzamide
methyl (2S,4S)-1-[1-(2-phenylethyl)piperidin-4-yl]-4-(thiophene-2-amido)pyrrolidine-2-carboxylate
[4-({4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}sulfamoyl)phenyl]urea
ethyl 4-[8-methyl-2-oxo-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinolin-4-yl]-1H-pyrazole-3-carboxylate
5-(4-acetylphenoxymethyl)-N-[(3-methylpyridin-4-yl)methyl]-1,2-oxazole-3-carboxamide
(3R,4R)-3-cyclopropyl-4-methyl-1-(5-methylthiophene-2-carbonyl)pyrrolidin-3-ol
3-{[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methyl}-2-methoxy-6-(propan-2-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-[1'-(2,6-dimethylpyrimidine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
ethyl 4-[(4-chlorophenyl)methyl]-1-ethylpiperidine-4-carboxylate
1-(2-{[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]methyl}morpholin-4-yl)ethan-1-one
(4aS,7aR)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{[3-(morpholin-4-yl)phenyl]methyl}-7-propyl-2,7-diazaspiro[4.5]decan-6-one
1-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-5-phenyl-1,2-oxazole
1-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}ethan-1-one
N-(1-{[ethyl(oxolan-2-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-3-(2-methoxyphenyl)propanamide
2-[(4-chlorophenyl)methyl]-8-(thiophen-3-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
6-(4-chlorophenyl)-N-methyl-N-(oxan-4-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(3-chlorophenyl)-7-fluoro-3-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}quinoline
3-{2-[cyclohexyl(methyl)amino]ethyl}-8-(oxolan-3-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-3-(1-oxo-2,3-dihydro-1H-inden-5-yl)urea
4-fluoro-N-[(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-3-yl)methyl]benzamide
1-{1,6-dimethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-(3-hydroxyquinoxalin-2-yl)propan-1-one
N-(2,3-dihydro-1H-inden-1-yl)-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
2-ethyl-4-methyl-N-[1-methyl-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]-1,3-oxazole-5-carboxamide
N-(2-ethylphenyl)-1-methyl-5-oxo-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
2-({[2-(morpholin-4-yl)ethyl]amino}methyl)-4-(pyrimidin-2-yl)phenol
2,5-dimethyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine