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(3S,7S)-5-[4-(1H-pyrazol-4-yl)butanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-(1,2-oxazol-3-ylmethyl)-7-(pyridazine-3-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{[2-(1H-indazol-6-yl)phenyl]methyl}dimethylamine
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
N-{2-[(2S)-2-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-2-carboxamide
N-methyl-2-[4-(pyrimidin-2-yl)piperazin-1-yl]-N-[1-(1,3-thiazol-5-yl)ethyl]acetamide
9-[(2-butyl-1H-imidazol-4-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
5-(6-methoxypyridazin-3-yl)-1H-indole
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
2-benzyl-4-[(1-methyl-1H-pyrazol-4-yl)methyl]morpholine
2-(5-acetylthiophen-3-yl)-N-[3-(methylamino)propyl]acetamide
1-[3-(3-fluorophenyl)phenyl]-3-[1-(hydroxymethyl)cyclopentyl]urea
1-[(2,3-difluorophenyl)methyl]-3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
4-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-chloro-N-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-4-fluoro-1-benzothiophene-2-carboxamide
2-(3-chloro-4-hydroxyphenyl)-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
(1S,5R)-3-[(2,3-difluorophenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 2-(azepane-1-sulfonyl)-6-(1,2,3-thiadiazole-4-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(pyrrolidine-1-carbonyl)pyrazin-2-amine
6-({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
N-methyl-3-[(5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)methyl]-1,2,4-oxadiazole-5-carboxamide
5-chloro-6-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyridine-3-carboxylic acid
5-fluoro-N4,N4-dimethyl-N2-[2-(pyrazin-2-yl)ethyl]pyrimidine-2,4-diamine
4-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-1-(propan-2-yl)piperidine
(2,1,3-benzoxadiazol-4-ylmethyl)(ethyl)({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)amine
5-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-2-methylphenol
4-(3-chlorophenoxy)-1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
2-methyl-4-(4-{3-[2-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}phenyl)but-3-yn-2-ol
methyl(pyrazin-2-ylmethyl){[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
1-(2-methylphenyl)-4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)-1,4-diazepane
3-[(methylamino)methyl]-4-(thiophen-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1R,9S)-5-amino-12-cyclopentyl-3-[5-(hydroxymethyl)furan-2-yl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-(1-{7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-phenylpropanamide
3-(1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)propan-1-ol
2-(cyclopropylmethyl)-8-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
2,4-dimethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyrimidine-5-carboxamide
N-({1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}methyl)-3-(trifluoromethyl)benzamide
4,5-dimethyl-6-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyrimidine
[(3-ethyl-1,2-oxazol-5-yl)methyl][(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]methylamine
1-{2-methyl-5-[2-(4-methylpentyl)morpholine-4-carbonyl]phenyl}imidazolidin-2-one
N-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)ethyl]-4-sulfamoylbenzamide
1-(cyclohex-1-en-1-ylmethyl)-3-(3-methanesulfonamido-4-methoxyphenyl)urea
N,1-dimethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)cyclohexane-1-carboxamide
6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-3-carboxamide
2-amino-7-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-3-(2-methylphenyl)-3-phenylpropanamide
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-N-ethylpyrimidin-2-amine
9-(2-hydroxybutanoyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-3,3-dimethylcyclohexan-1-amine
4-(2-methylpyrrolidine-1-carbonyl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline