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1-phenyl-4-[2-(2,2,6,6-tetramethylpiperidin-4-yl)acetyl]piperazin-2-one
3,5-dichloro-4-methyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]benzamide
1-[3-(2,3-dihydro-1,4-benzodioxin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N-[3-(furan-2-yl)phenyl]-1-(1,2,5-thiadiazole-3-carbonyl)piperidine-4-carboxamide
9-(3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
(1S,5R)-3-{[3-(benzyloxy)phenyl]methyl}-3,9-diazabicyclo[3.3.2]decan-10-one
5-phenyl-N-[(3R)-pyrrolidin-3-yl]-1,2-oxazole-4-carboxamide
6-(4-fluorophenyl)-3-(2-methoxyethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
4-(2,3-dimethyl-1H-indole-5-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2-[4-(dimethylcarbamoyl)phenyl]-2-[(isoquinolin-5-ylmethyl)(methyl)amino]acetic acid
4-[(2,3-difluoro-6-methoxyphenyl)methyl]-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
2-(2-methoxyethyl)-8-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)-2-ethyl-2,5-dihydro-1H-pyrrole-1-carboxamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-(quinolin-4-yl)piperazin-2-yl}ethan-1-ol
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1,2-oxazole-3-carboxamide
[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
3-[1-(4-cyanopyridin-2-yl)piperidin-3-yl]-N-[(3,4-difluorophenyl)methyl]propanamide
2-(3-methyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
6-[2-(3,4-dichlorophenyl)morpholin-4-yl]-N,N-dimethylpyridine-3-carboxamide
N-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-4-(2-methylpyridin-4-yl)piperazine-1-carboxamide
8-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
8-{2-[5-(dimethyl-1,2-oxazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethoxy}quinoline
3-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridazine
methyl({[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl})[1-(1,2-oxazol-3-yl)ethyl]amine
1-(propane-2-sulfonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-[(4,6-dimethylpyridin-3-yl)methyl]-6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[1-(1H-imidazol-2-yl)ethyl]-7-[(4-methyl-1H-imidazol-5-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-({1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-2-yl}methyl)morpholine
1-ethyl-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
5-methyl-2-[3-(pyridin-3-ylmethyl)-1,2,4-oxadiazol-5-yl]-1H-indole
(1R,2S,9R)-11-(2,1,3-benzoxadiazol-4-ylmethyl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
methyl 2-({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-1,3-oxazole-4-carboxylate
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-4-carboxamide
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-4-propylpyrimidine-5-carboxamide
[2,4,6-trimethyl-3-({[1-(1-methyl-1H-pyrazol-5-yl)propyl]amino}methyl)phenyl]methyl acetate
5-methyl-1-{2-[3-(oxan-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1-(1-methyl-1H-imidazole-5-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
1-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}-4-(propan-2-yl)piperazine
2-methyl-6-(1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)pyrimidin-4-ol
methyl 6-[(4-chlorophenyl)methyl]-2-[(2-methoxyethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl 3-[(2R)-2-carbamoylpyrrolidine-1-carbonyl]-5-(cyclobutylmethoxy)benzoate
3-(hydroxymethyl)-N-(3-methoxyphenyl)-3-[(2-methylphenyl)methyl]piperidine-1-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}propanamide
1-[3-(1,3-benzothiazol-2-yl)propyl]-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)urea
5-tert-butyl-3-{[3-(4-methylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-pyrazole
1-[(5-ethylfuran-2-yl)methyl]-3-(3-methylthiophene-2-carbonyl)piperidine
4-phenyl-1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrrolidin-2-one
N-[(3S,4R)-1-(3-chloropyridin-2-yl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide