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N-(pyridin-3-ylmethyl)-4-{[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]amino}pyridine-2-carboxamide
3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-8-[(4-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-methyl-2-({3-[2-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(pyrazin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-(piperidin-4-yl)acetamide
2-methyl-5-(4-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}phenyl)-2H-1,2,3,4-tetrazole
[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
5-(4-fluorophenyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
3-methyl-1-(2-oxo-2-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}ethyl)-1,2,3,4-tetrahydroquinazolin-2-one
1-[2-(dimethylamino)-4-({3-[(pyridin-3-yl)amino]propyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-(2,3-dimethylquinoxalin-6-yl)-3-(3-hydroxypropyl)-3-(thiophen-2-ylmethyl)urea
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)pyrrolidine-1-carboxamide
2-{1-cyclopentyl-4-[4-(1,2,4-oxadiazol-3-yl)pyridin-2-yl]piperazin-2-yl}ethan-1-ol
7-fluoro-3-methyl-2-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-indole
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-3-(dimethyl-1,2-oxazol-4-yl)propanamide
8-[2-(2-oxopyrrolidin-1-yl)acetyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-[(3-ethoxyphenyl)methyl]-1-(2-hydroxyethyl)urea
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
(1R,3S)-7-[(3-chloro-1-benzothiophen-2-yl)methyl]-7-azaspiro[3.5]nonane-1,3-diol
N-(1,3-dihydroxy-2-methylpropan-2-yl)-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]-2-(1-methyl-1H-pyrazol-4-yl)quinoline
N-{1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}pyridine-3-carboxamide
(1S,3R)-N-ethyl-2,2,3-trimethyl-3-[4-(prop-2-en-1-yl)piperazine-1-carbonyl]cyclopentane-1-carboxamide
6-cyclopentyl-N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2R,3R)-3-amino-1'-(3-fluoro-4-methylbenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-(dimethylamino)-3-[4-({methyl[2-(4-methylphenoxy)ethyl]amino}methyl)phenoxy]propan-2-ol
2-(3-hydroxypropyl)-9-(1,3-thiazol-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(2H-1,3-benzodioxol-5-yl)-3-(thiomorpholin-4-yl)-1,2,4-triazine
3-methyl-1-(2-{9-oxa-2-azaspiro[5.5]undecan-2-yl}-2-oxoethyl)-1,2-dihydroquinoxalin-2-one
2-{[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]amino}-N-(1,3-thiazol-2-yl)propanamide
6-methoxy-3-methyl-N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
4-{1-[1-(pyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-[(pyridin-2-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
2-(2-{[6-hydroxy-4-(2-hydroxyethyl)-1,4-diazepan-1-yl]methyl}phenoxy)acetic acid
(1S,4S)-2-(2-chlorophenyl)-5-[4-(trifluoromethyl)benzoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
(2S,4S)-N-(2-phenylethyl)-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
3-chloro-4-({2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}sulfonyl)benzonitrile
1-(3-butoxyphenyl)-3-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-3-methylurea
3-(3,5-dimethylphenyl)-N-[(4-sulfamoylphenyl)methyl]propanamide
6-methyl-N4-{3-[(5-methylpyridin-2-yl)amino]propyl}pyrimidine-2,4-diamine
2-(4-fluorophenyl)-N-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)morpholine-4-carboxamide
({4-cyclopropyl-5-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-[(2-methoxyphenyl)methyl]-4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
2-ethoxy-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)acetamide
4-(4-chloro-1H-pyrazole-3-carbonyl)-1-(cyclopropylmethyl)-2-(propan-2-yl)-1,4-diazepane
1-methyl-5-[4-(4-phenylpyrimidin-2-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide