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N-[2-(6-methylpyridin-2-yl)ethyl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
1-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-5-yl]urea
(2S,4R)-4-(dimethylamino)-1-[2-(phenylsulfanyl)acetyl]pyrrolidine-2-carboxylic acid
1-cyclopentyl-N3-methyl-N3-(2-methylpropyl)-4-oxo-N5-[1-(thiophen-3-yl)propan-2-yl]-1,4-dihydropyridine-3,5-dicarboxamide
4-[(3-methoxyphenyl)methyl]-11-[(2-methylpropyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[(2-chlorophenyl)methyl]-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-[4-(2-ethyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidine-1-carbonyl]quinoline
N-(3-hydroxypropyl)-1-{1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
(1R,5S,6R)-3-(1H-1,3-benzodiazol-2-ylmethyl)-N-[(3-methylphenyl)methyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide
2-{2-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethoxy}acetamide
1-{9-[(3-ethenylphenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl}-2-methoxyethan-1-one
7-(2-cyclohexylethyl)-2-(pyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decane
1-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
4-[1-benzyl-5-(4,4,4-trifluorobutan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
4-ethyl-1-[(2E)-3-phenylprop-2-en-1-yl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-2H-1,3-benzodioxole-5-carboxamide
6-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridin-3-ol
3-[4-(2-methylpyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridine
5-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)-4-ethyl-1,2,3-thiadiazole
1-(2H-1,3-benzodioxol-4-ylmethyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(3-hydroxy-3-methylbutyl)benzamide
3-{[(1R)-1-(2-fluorophenyl)ethyl]sulfamoyl}-N-[2-(methylamino)ethyl]benzamide
2-[(3-methoxyphenyl)methyl]-8-[3-(methylsulfanyl)butyl]-2,8-diazaspiro[4.5]decan-3-one
dimethyl({4-[1-(quinoline-6-carbonyl)piperidin-2-yl]phenyl}methyl)amine
ethyl 4-(2-phenoxyethyl)-1-(pyridin-2-ylmethyl)piperidine-4-carboxylate
1-(4-methoxyphenyl)-4-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]butane-1,4-dione
methyl 4-(6-chloro-2H-chromen-3-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylate
N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-(5-methyl-1,2-oxazol-3-yl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidine
5-(2-methylpropyl)-3-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1H-pyrazole
4-(cyclopropylmethyl)-1-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-cyclohexyl-4-[2-(1H-1,2,4-triazol-5-yl)benzoyl]piperazin-2-one
methyl 3-benzamido-5-{[(3-methylthiophen-2-yl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-cyclopentanecarbonyl-N-[3-(pyridin-2-yl)propyl]piperidine-4-carboxamide
7-[(3,4-difluorophenyl)methyl]-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(furan-3-ylmethyl)(methyl)[(3-{[1-(4-phenylbenzoyl)piperidin-4-yl]oxy}phenyl)methyl]amine
2-{[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]oxy}-N-cyclopropyl-4-methoxybenzamide
4-[1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]benzoic acid
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-6-ethyl-N-methyl-2-(morpholin-4-yl)pyrimidin-4-amine
3-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-N-(1H-pyrazol-3-ylmethyl)benzene-1-sulfonamide
8-(1,3-benzothiazol-2-ylmethyl)-3-benzyl-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
4-(3-methylpyridine-2-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{1-cyclohexyl-4-[(3,4-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-ethyl-6-{[2-(1H-imidazol-4-yl)ethyl]amino}-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
methyl (2S)-1-[2-(morpholin-4-yl)-6-phenylpyridine-3-carbonyl]pyrrolidine-2-carboxylate
(4aR,7aS)-1-methyl-4-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
methyl (2S)-1-[9-methoxy-7-oxo-3-(3-phenylprop-2-ynoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]pyrrolidine-2-carboxylate
N-(1-benzothiophen-2-ylmethyl)-N-methyl-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide