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5-[({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]pyrimidin-2-amine
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-2-(morpholin-2-yl)ethan-1-one
2-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-6-(trifluoromethyl)pyridine-3-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-{[4-(methylsulfanyl)phenyl]carbamoyl}piperidine-4-carboxylate
4-amino-1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-3-hydroxybutan-1-one
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidine
3-[(3,4-dimethoxyphenyl)methyl]-N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
7-(cyclopropylmethyl)-2-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}-N-(pyrrolidin-3-yl)benzamide
4-[2-(2-chloro-4-fluorophenoxy)propanoyl]-1-phenylpiperazin-2-one
N3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-methoxy-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-[3-(methylsulfanyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
methyl[(1-methyl-1H-indol-3-yl)methyl][1-(pyridin-2-yl)ethyl]amine
N-(propan-2-yl)-3-{5-[2-(1H-pyrazol-1-ylmethyl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,2,3-benzotriazole-5-carboxamide
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(2,2,2-trifluoroethyl)piperazin-1-yl]ethan-1-one
7-(1-benzothiophen-3-yl)-4-[(2-methyl-1H-imidazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(azepan-1-yl)-3-[3-({[(2-chlorophenyl)methyl]amino}methyl)phenoxy]propan-2-ol
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(methylsulfanyl)phenyl]urea
N-cyclooctyl-3-[4-(2-ethoxyethyl)piperazin-1-yl]propanamide
N-(2,4-dimethoxyphenyl)-3-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}propanamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]acetamide
1-(2-methoxy-4-{[(2-phenoxyethyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
N-ethyl-4-(1-phenyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-{[(3S)-3-(dimethylamino)pyrrolidin-1-yl]methyl}-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
1-[2-(dimethylamino)ethyl]-N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
7-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2-oxa-7-azaspiro[4.5]decane
N-[(3R,4R)-3-hydroxy-1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-4-yl]pyrazine-2-carboxamide
8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({7-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenylacetamide
5-[3-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
3-[ethyl(pyridin-4-ylmethyl)amino]-N-(4-methoxyphenyl)piperidine-1-carboxamide
N-(1-{1-[(3-ethoxy-2-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
5-(2-cyclopentylacetamido)-N-(2,3-dihydro-1H-inden-2-yl)-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
2-{4-[1-(2-hydroxybutyl)-1H-1,2,4-triazol-5-yl]phenoxy}acetamide
(3S)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-N,N-dimethylazepan-3-amine
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-1,2,5-oxadiazole-3-carboxamide
3-{[ethyl(methyl)amino]methyl}-4-(5-fluoro-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-ethyl-N,2,3-trimethyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(3-methoxyphenyl)-4-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)benzamide
8-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-ethyl-1-methyl-N-(pyridin-4-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
3-[(2-fluorophenyl)formamido]-N-[2-(N-methylmethanesulfonamido)ethyl]propanamide
4-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
(3R)-3,4,4-trimethyl-1-{5-[(4-methylpiperazin-1-yl)methyl]furan-2-carbonyl}pyrrolidin-3-ol
5-({[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]amino}methyl)pyrrolidin-2-one