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3-(4-phenoxybenzoyl)-1-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperidine
1'-(1,3-thiazol-2-yl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetamide
2-(3,5-dichloropyridin-4-yl)-1-methyl-1H-1,3-benzodiazole
N-[(1-methyl-3-phenyl-1H-pyrazol-5-yl)methyl]-6-(morpholin-4-yl)pyrimidin-4-amine
4-(2-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-2-yl}ethyl)morpholine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-2H-1-benzopyran-2-carboxamide
methyl(quinolin-6-ylmethyl){[4-(2-{4-[2-(trifluoromethyl)benzenesulfonyl]piperazin-1-yl}ethoxy)phenyl]methyl}amine
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)cyclohexanecarboxamide
4-(4-ethoxy-3-methylphenyl)-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4-oxobutanamide
2-(2,4-dioxoimidazolidin-1-yl)-N-[(3R,4S)-4-propyl-1-(1,3-thiazol-2-yl)pyrrolidin-3-yl]acetamide
1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-4-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1,4-diazepan-2-one
1-[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]-2,2-dimethylpropan-1-one
6-[2-(pyridin-4-yl)-1H-imidazol-1-yl]-1H-indazole
5-cyclopentyl-3-({5-[2-(methylsulfanyl)propyl]-4-phenyl-1H-imidazol-1-yl}methyl)-1,2,4-oxadiazole
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
2-ethyl-8-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-2,8-diazaspiro[5.5]undecane
6-amino-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)pyridine-3-carboxamide
1-(3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-3-(2-methylphenyl)propan-1-one
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(6-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetamide
1-[4-(3-aminopyrrolidin-1-yl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
7-chloro-3,5-dimethyl-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-benzofuran-2-carboxamide
3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}quinoxaline-5-carboxamide
1-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
5-(1-{[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-N,N-dimethylthiophene-2-carboxamide
ethyl 1-[2-(methylsulfamoyl)ethyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
2-chloro-N-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}-3-methylbenzamide
N-cyclopropyl-N-({4-[3-(dimethylamino)propoxy]phenyl}methyl)cyclohexanecarboxamide
2-(1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
1-methyl-3-{3-[4-(3-propylpyrrolidin-1-yl)piperidin-1-yl]phenyl}imidazolidin-2-one
3-(3-hydroxy-3-methylbutyl)-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}benzamide
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-4-(N-methylmethanesulfonamido)benzamide
N-{[3-(dimethylamino)thiolan-3-yl]methyl}-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
(3S,4R)-3-benzyl-1-(3-hydroxybenzoyl)-4-methylpiperidin-4-ol
N-[(3-chlorophenyl)methyl]-N-propyl-3-(1H-pyrazol-1-yl)butanamide
6-(4-chlorophenyl)-N-[(3-methylpyridin-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[2-(2,4-difluorophenyl)pyridine-4-carbonyl]-4-methylpiperazine
N,N-dimethyl-2-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]aniline
1-(2-cyclopropylpyrimidine-5-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-{2-oxo-2-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethyl}piperazin-2-one
1-{2-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-oxoethyl}azepan-2-one
2-[5-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)furan-2-yl]benzonitrile
N-(3-methoxypropyl)-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-(2,3-difluorophenyl)-4-[(2-ethyl-1H-imidazol-1-yl)methyl]-5-methyl-1,3-oxazole
9-(dimethoxy-1,3,5-triazin-2-yl)-3-oxa-9-azaspiro[5.5]undecane
3-chloro-4-{[2-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}pyridine
(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)-N-[2-(trifluoromethyl)phenyl]pyrrolidine-1-carboxamide