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1-[(4-methylphenyl)amino]-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]cyclopentane-1-carboxamide
2-{[2-(2,5-dimethylphenyl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-6-methylimidazo[1,2-a]pyridine-2-carboxamide
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}amine
1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
1-ethyl-4-({methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]amino}methyl)-1H-pyrrole-2-carbonitrile
N-(furan-2-ylmethyl)-N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
3-[1-(quinoline-8-carbonyl)piperidin-3-yl]benzoic acid
8-(3-chloropyridin-2-yl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-(2,5-dimethylfuran-3-carbonyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[3-(methylsulfanyl)propyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,1-dimethyl-1H-pyrazole-5-carboxamide
methyl({[4-(5-methylfuran-2-yl)phenyl]methyl})(1,2-oxazol-3-ylmethyl)amine
1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]ethan-1-one
2-(1-{[1-(2-ethylpyrimidine-5-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
(4aR,7aS)-1-propanoyl-4-(pyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl({[(1R,5S,6R)-3-(2-methylbenzoyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl})[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
5-{4-[(4-chlorophenyl)methyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-[(3-propyl-1,2-oxazol-5-yl)methyl]urea
1-[(4-hydroxy-3-methoxyphenyl)methyl]-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-methyl-5-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-cyclohexanecarbonyl-7-[2-methyl-2-(morpholin-4-yl)propyl]-2,7-diazaspiro[4.5]decane
5-[(4-cyclobutanecarbonyl-1,4-diazepan-1-yl)methyl]-2-hydroxybenzoic acid
N-{[1-(pyridazine-4-carbonyl)piperidin-3-yl]methyl}naphthalene-1-carboxamide
N-(2-methylpropyl)-5-(morpholin-4-ylmethyl)-N-(thiophen-3-ylmethyl)furan-3-carboxamide
3-hydroxy-3-{[(2-methylbutan-2-yl)amino]methyl}-1-(3-phenylpropyl)piperidin-2-one
4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-(pyridin-3-yl)morpholine
N3-(1,3-benzothiazol-2-ylmethyl)-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methoxypropan-1-one
N-cyclopropyl-3-[5-(6-methyl-2-propylpyrimidin-4-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
1-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidin-2-one
2-{4-[(5-chlorothiophen-2-yl)methyl]morpholin-3-yl}-N-(cyclohex-1-en-1-ylmethyl)acetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(3-methylthiophen-2-yl)methyl]piperidin-3-ol
2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethan-1-one
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]propanamide
N-({3-methyl-7-[2-(methylsulfanyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(piperidin-1-yl)acetamide
3-benzyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[4-(4-chloro-2-hydroxybenzoyl)piperazin-1-yl]-1-(piperidin-1-yl)ethan-1-one
3-(4-ethylphenyl)-5-[(4-methanesulfonylphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-N'-(4-methylpyridin-2-yl)butanediamide
1,3-dimethyl-4-[1-(thiophene-2-carbonyl)piperidin-4-yl]piperazin-2-one
2-(carbamoylamino)-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}acetamide
N-[(3R,4R)-3-hydroxy-1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-4-yl]pyridine-2-carboxamide
(1R,3S,5S)-8-({5-[(3-hydroxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-8-azabicyclo[3.2.1]octan-3-ol
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(phenylsulfanyl)ethan-1-one
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chlorophenyl)urea
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
methyl 4-{[3-(benzylcarbamoyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}benzoate
4-[1-(2-phenylethyl)-5-(5-propyl-1,2-oxazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine