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N-(3,4-dihydro-2H-1-benzopyran-3-yl)-5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
2-{3-cyclopropyl-5-[4-(2-methoxyphenyl)phenyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
4-cyclopentyl-6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-hydroxy-1-[6-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
(3S,4S)-1-{[4-(2-methylpropyl)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
(5S)-5-[3-(3-chlorophenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidin-2-one
(3S,4S)-4-cyclopropyl-1-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrrolidine-3-carboxylic acid
N-benzyl-N-cyclopentyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
4-oxo-4-{4-oxo-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}butane-1-sulfonamide
1-{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(oxolan-2-yl)-1H-1,3-benzodiazole
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(4-methylpent-3-en-1-yl)pyrrolidin-3-yl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-5-methoxyfuran-2-carboxamide
3-[3-(1-methylpiperidin-4-yl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
3-(dimethyl-1,2-oxazol-4-yl)-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)propan-1-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-4-methyl-N-(2-methylpropyl)-1,3-thiazole-5-carboxamide
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3-(3-methylphenyl)piperidine
5-methyl-1'-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]({[5-(methoxymethyl)furan-2-yl]methyl})methylamine
(4aS,8aR)-1-(4-hydroxybutyl)-6-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
ethyl 4-{4-[(2-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}piperidine-1-carboxylate
1-(4,6-dimethoxypyrimidin-2-yl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-benzyl-4-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazin-2-one
3-(3-methylbutyl)-8-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N'1-[(1-ethylpyrrolidin-2-yl)methyl]-N'1-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}cyclopropane-1,1-dicarboxamide
2-(4-chloro-2-{[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]methyl}phenoxy)acetic acid
(2S,4S)-4-amino-1-{[2,5-dimethyl-1-(4-methylpyridin-2-yl)-1H-pyrrol-3-yl]methyl}-N-methylpyrrolidine-2-carboxamide
2-(4-{[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]methyl}phenyl)acetic acid
(2S,4S)-4-(3,6-dimethyl-1-benzofuran-2-amido)-1-methylpyrrolidine-2-carboxylic acid
1-(2-{[(1S,2S)-2-(benzyloxy)cyclohexyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one
2-(2,3-dihydro-1H-inden-1-yl)-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)acetamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]ethan-1-one
4-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-2-(trifluoromethyl)morpholine
[1-(1,3-benzothiazol-2-ylmethyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
3-(1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-yl)propan-1-ol
1-(4-{[4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)propan-1-one
2-{2-chloro-4-[(3-propoxypiperidin-1-yl)methyl]phenoxy}acetamide
N-[2-(2-chlorophenyl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
4-(3-fluoropyridin-4-yl)-7-phenoxy-1,2,3,4-tetrahydroquinolin-2-one
1-(4-aminopyridine-2-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
[(3R,5R)-5-[(dimethylamino)methyl]-1-(3-methoxybenzoyl)piperidin-3-yl]methanol
4-ethyl-1-methyl-3-[(1-{[2-(propylamino)pyrimidin-5-yl]methyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[4-(2-fluoro-6-methoxybenzoyl)-2-oxopiperazin-1-yl]benzonitrile
(2S)-N-{3-[ethyl(phenyl)carbamoyl]phenyl}-5-oxopyrrolidine-2-carboxamide
N,N-dimethyl-2-[(1S,5R)-3-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-2,6-dimethylquinoline-4-carboxamide
3-chloro-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]thiophene-2-carboxamide
7-(1-benzothiophen-3-yl)-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-9-[2-(pyridin-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-1-(morpholin-4-yl)propan-1-one