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2-cyclopentyl-1-{4-[4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}-2-phenylethan-1-one
4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]piperazine-2-carboxylic acid
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-[2-(6-methylpyridin-2-yl)ethyl]pyridin-2-amine
1-{2-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(5-{[4-(oxolane-2-carbonyl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
1-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
4-{[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}phenol
N-(2-methoxyethyl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-(propan-2-yl)acetamide
6-methyl-5-[5-(1-methylpiperidin-4-yl)-1,2,4-oxadiazol-3-yl]-2-(pyrazin-2-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
N-(1-benzothiophen-5-ylmethyl)-2-(morpholin-2-yl)acetamide
5-{[5-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-3-ethyl-4,5-dihydro-1,2-oxazole
N-[4-(3-fluorophenyl)phenyl]-1-(thian-4-yl)piperidine-3-carboxamide
N-[4-({[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]carbamoyl}methoxy)phenyl]propanamide
1-methyl-N-(2-phenylethyl)-N-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}piperidin-4-amine
1-(2-aminoethyl)-N-[2-(4-fluorophenyl)ethyl]-N-(pyridin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(3-methoxypropyl)-N-{[2-(3-methylphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}furan-3-carboxamide
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N,1-dimethyl-1H-indole-2-carboxamide
N-methyl-5-(propan-2-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,2-oxazole-3-carboxamide
N-(2,4-dimethoxyphenyl)-3-[1-(4-phenylbutan-2-yl)piperidin-4-yl]propanamide
2-amino-4-(1,3-dimethyl-1H-pyrazol-4-yl)-6-[4-methyl-2-(piperidin-1-yl)pyrimidin-5-yl]pyridine-3-carbonitrile
6-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-hydroxypropanamide
(3S,4R)-1-[(3-fluoro-4-methoxyphenyl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
1-(3-chlorophenyl)-4-[2-(dimethylamino)acetyl]-5-methylpiperazin-2-one
ethyl 3-[(3-chlorophenyl)methyl]-1-(2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetyl)piperidine-3-carboxylate
3-[4-(dimethylamino)phenyl]-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]propan-1-one
1-{2-oxo-2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{2-[1-(quinolin-2-ylmethyl)piperidin-3-yl]ethyl}methanesulfonamide
N-[3-(1H-indol-2-yl)phenyl]-1-(pent-4-enoyl)piperidine-4-carboxamide
3-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
N-(cyclohex-1-en-1-ylmethyl)-3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)propanamide
N-(propan-2-yl)-1-[1-(quinoline-8-sulfonyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
8-[6-(piperidine-1-carbonyl)pyrazin-2-yl]quinoline
4-{3-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]propoxy}benzamide
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl){[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amine
N-[(4-fluorophenyl)methyl]-3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
2-(3-chloropyridin-2-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
1-{1-[6-(aminomethyl)-2-methylpyrimidin-4-yl]piperidin-4-yl}piperidin-3-ol
(4aS,8aR)-6-(2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
8-{5-[(4,5-dimethylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}quinoline
4-(4,4-difluoropiperidine-1-carbonyl)-6-ethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
methyl 3-(2-chlorobenzamido)-5-[(cyclopropylformamido)methyl]benzoate
(1R,5S,8R)-N,N-dimethyl-3-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-3-azabicyclo[3.2.1]octan-8-amine
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
N-methyl-N-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
3,5-dimethyl-N-(oxan-2-ylmethyl)-1-benzofuran-2-carboxamide
N-[4-methoxy-3-(methylcarbamoyl)phenyl]-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-(4-cyclopentyl-1,4-diazepan-1-yl)butan-1-one
4-(2-acetylbenzoyl)-6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one