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(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-6-(morpholine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}-N-(1,3-thiazol-2-yl)propanamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
1-[(2,5-dimethylphenyl)methyl]-4-[2-(4-methyl-1,4-diazepane-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
1-{3-[4-(morpholine-4-carbonyl)pyridin-2-yl]phenyl}ethan-1-one
(3aR,6aR)-2-cyclobutanecarbonyl-5-(2-fluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(2-methoxyethyl)-3-propyl-1-(4-sulfamoylphenyl)urea
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
methyl 2-(2-{[(2S)-2-acetamidopropanamido]methyl}-5-methyl-2,3-dihydro-1-benzofuran-7-yl)benzoate
4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-[(3,5-dimethoxyphenyl)methyl]piperidine
ethyl 3-benzyl-1-(ethanesulfonyl)piperidine-3-carboxylate
(3S,4S)-1-(4-methylpyrimidin-2-yl)-4-(naphthalen-2-yl)piperidin-3-ol
N-[(4-methyl-1H-imidazol-2-yl)methyl]-3-(pyridin-3-yl)propanamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
N-[3-(azepan-1-yl)propyl]-N-methylfuran-3-carboxamide
9-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-5-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1H-1,2,3-benzotriazole
7-methoxy-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-methoxy-1-(4-{2-[(1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]phenoxy}piperidin-1-yl)ethan-1-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-(5-methylpyridine-2-carbonyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(1S,4S)-2-(2-fluorophenyl)-5-[(1-methyl-1H-indol-3-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
4-(1H-imidazol-2-yl)-1-[4-(trifluoromethyl)benzoyl]piperidine
N-[(2-fluorophenyl)methyl]-3-[1-(furan-2-carbonyl)piperidin-3-yl]propanamide
2,6-dimethyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}quinoline-4-carboxamide
1-{2-[2-(dimethylamino)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-2-(furan-2-yl)ethane-1,2-dione
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-2-(pyridin-3-yloxy)acetamide
1-(4,6-dimethylpyrimidin-2-yl)-N-[1-(pyrimidin-4-yl)ethyl]piperidin-4-amine
2-chloro-N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-5-(trifluoromethyl)benzamide
2-{4-[4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carboxamide
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
3-[(2,1,3-benzoxadiazol-5-ylmethyl)sulfamoyl]-N-[2-(methylamino)ethyl]benzamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
1-{1-[6-(2,5-difluorophenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
(2R,3R)-3-amino-1'-[(3-chloro-4-fluorophenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(1H-imidazol-2-ylmethyl)({[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl})methylamine
N-[1-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
(2S,4R)-N-ethyl-4-(2-methylfuran-3-amido)-1-(thiophen-2-ylmethyl)pyrrolidine-2-carboxamide
2-amino-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-phenylpyrimidine-5-carboxamide
3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-methylpyridine
1-[(3S,4R)-4-ethoxyoxolan-3-yl]-5-(1-ethyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazole
(4-{[methyl({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}oxan-4-yl)methanol
N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
(4aS,8aR)-6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-(1,4-dioxan-2-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl][1-(2,6-dimethylphenoxy)propan-2-yl]amine
1-(1-{6-[(3-hydroxypropyl)amino]pyridine-3-carbonyl}piperidin-3-yl)-3-methylbutan-1-one