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[3-(2-{[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]amino}ethyl)-1,2,4-oxadiazol-5-yl]methanol
(4aS,8aR)-6-[(2-aminopyridin-3-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2,2-dimethyloxan-4-amine
N-methyl-N-(2-phenyl-1-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}ethyl)pyridine-2-carboxamide
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-3-ethoxypropan-1-one
ethyl 2-[1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidin-2-yl]acetate
N-[3-(cyclohexyloxy)propyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
4-[(4-fluorophenyl)methyl]-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-[2-(1-methylpiperidin-3-yl)ethyl]-2-(1,2,3,6-tetrahydropyridin-4-yl)acetamide
2-(2-hydroxyethyl)-8-{2-[4-(hydroxymethyl)phenyl]acetyl}-2,8-diazaspiro[5.5]undecan-3-one
N-(1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
ethyl 1-[5-(3-acetylphenoxymethyl)-1H-pyrazole-3-carbonyl]piperidine-3-carboxylate
(1S,5R)-3-(5-acetylpyridin-2-yl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
9-hydroxy-2-{[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]methyl}-4H-pyrido[1,2-a]pyrimidin-4-one
1-[(3S)-3-ethylmorpholin-4-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
5-{1-[(4-chlorophenyl)methyl]-4-hydroxypiperidin-4-yl}-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1-benzofuran-2-carboxamide
(6-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}pyridin-2-yl)methanol
1-(cyclohex-3-ene-1-carbonyl)-3-phenylpyrrolidin-3-ol
[(4-{[1-(furan-3-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
3-benzoyl-1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
4-methyl-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-(azepan-1-yl)-3-(4-chloro-2-{[(3-hydroxypropyl)(methyl)amino]methyl}phenoxy)propan-2-ol
1-(3-fluorobenzoyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-methyl-N-[2-(7-methyl-1H-indol-3-yl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-{2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}-1H-indole
1-ethyl-N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-(3,5-dichloro-4-methylbenzoyl)-1,4-oxazepane
N-[(1S,2R)-2-aminocyclobutyl]-2-methyl-5-(2-methyl-1,3-oxazol-5-yl)benzene-1-sulfonamide
4-[(dimethylamino)methyl]-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]azepan-4-ol
2-(2H-1,3-benzodioxol-5-yloxy)-1-[4-(dimethylamino)azepan-1-yl]ethan-1-one
N-{4-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-4-oxobutyl}acetamide
4-(3,3-dimethylpyrrolidine-1-carbonyl)-7-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
N-[3-(pyridin-3-yloxy)propyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2-(2,5-dimethylphenoxy)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
6-methyl-3-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]pyrrolidin-3-yl]methanol
1-(5-chloro-2-fluorobenzoyl)-2-(3-methoxypropyl)piperidine
2-{[5-(oxan-4-yl)-4-phenyl-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
6-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-oxo-4H-pyran-2-carboxamide
(3R,4S)-1-{6-chloroimidazo[1,2-a]pyrimidine-2-carbonyl}-3,4-dimethylpiperidin-4-ol
1-[(4aR,8aS)-1-(2-methylbenzoyl)-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
2-methyl-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-(2,2-dimethyloxane-4-carbonyl)-4-{2-[(3-methoxyphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-[(2-fluorophenyl)methyl]-1,4-diazepane
[(3R,4R)-1-(2-amino-5,6,7,8-tetrahydroquinazoline-4-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
7-chloro-2-(2-methoxyphenyl)-3-(morpholin-4-ylmethyl)quinoline
3-[(2-methoxyethyl)sulfamoyl]-5-(quinolin-5-yl)benzoic acid
3-(3,4-dimethoxybenzoyl)piperidine
2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-N,N-diethylacetamide
5,6-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]thieno[2,3-d]pyrimidin-4-amine