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N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-cyclopropyl-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-[4-(hydroxymethyl)piperidin-1-yl]acetic acid
7-chloro-4-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-4H-pyrido[1,2-a]pyrimidin-4-one
4-{2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carbonyl}-3-ethylmorpholine
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)cyclohexanamine
3-(2H-1,3-benzodioxol-5-yl)-N-benzyl-N-(3-hydroxy-2-methylpropyl)propanamide
1-{[5-(oxan-2-yl)furan-2-yl]methyl}-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-2-(dimethylamino)-2-(3-methylphenyl)ethan-1-one
4-({1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidin-4-yl}methyl)morpholine
8-[3-(dimethylsulfamoyl)propyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[5-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
N-benzyl-5-(3,4-difluorophenoxymethyl)-N-ethyl-1,2-oxazole-3-carboxamide
N-methyl-2-(2-oxo-1,2-dihydroquinoxalin-1-yl)-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}acetamide
2-(2-ethoxyphenyl)-5-methyl-4-[(2-propyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
2-(cyclopropylmethyl)-5-[methyl(2-phenylethyl)amino]-2,3-dihydropyridazin-3-one
5-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
2-[(2-methylpyrimidin-5-yl)methyl]-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
N-ethyl-3-methyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}thiophene-2-carboxamide
N-(furan-2-ylmethyl)-N-(prop-2-en-1-yl)quinoline-3-carboxamide
1-[1-(3-hydroxy-4-methylbenzoyl)piperidin-3-yl]-3-phenylpropan-1-one
N-{[1-(carbamoylmethyl)-1,2,3,6-tetrahydropyridin-4-yl]methyl}-N-ethyl-2-phenylacetamide
N-{[4-(hydroxymethyl)phenyl]methyl}-3-(1-methyl-1H-pyrazol-4-yl)propanamide
7-[4-(4-propylphenyl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 3-[2-(1H-pyrazol-1-yl)acetamido]-5-({[2-(trifluoromethyl)phenyl]formamido}methyl)benzoate
3-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
1-{2-[3-(3-methylphenyl)piperidin-1-yl]-2-oxoethyl}piperidine-4-carboxamide
3-ethyl-N-({1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)-1,2-oxazole-5-carboxamide
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2,2-dimethyloxane-4-carboxamide
[(4-methanesulfonylphenyl)methyl](2-methoxyethyl)[(4-methylphenyl)methyl]amine
3-methyl-6-{5-[2-(4-methylbenzoyl)phenyl]-1,2,4-oxadiazol-3-yl}pyridazine
3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,4-dimethoxyphenyl)methyl]piperidine
5-cyclobutanecarbonyl-1'-(cyclohex-3-en-1-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(3-methoxypropyl)-3-(pyrimidin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3R,4S)-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3,4-dimethylpiperidin-4-ol
ethyl 4-[9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(1,4-dithiepan-6-yl)piperidine-3-carboxylate
3-(3-{[(2-methylpropyl)(thiophen-3-ylmethyl)amino]methyl}-1H-indol-1-yl)propanamide
2-methyl-8-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-(cyclopropylsulfamoyl)-5-(pyridin-3-yl)benzoic acid
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]acetamide
1-ethyl-6-methyl-2-oxo-N-[2-(4-sulfamoylphenyl)ethyl]-1,2-dihydropyridine-3-carboxamide
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-3-ethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
2-amino-4-(2-methoxypyrimidin-5-yl)-6-(1-methylcyclopropyl)pyridine-3-carbonitrile
N-[(2S)-1-methoxypropan-2-yl]-3-{[(2S)-pyrrolidin-2-ylmethyl]sulfamoyl}benzamide
N-{[6,7-dimethoxy-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-2-fluoro-N-(oxolan-2-ylmethyl)benzamide
5-[4-phenyl-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-imidazol-5-yl]pyrimidin-2-amine
1-[3-(7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)phenyl]imidazolidin-2-one
N-{[(2S,4S)-4-fluoro-1-(5-phenoxyfuran-2-carbonyl)pyrrolidin-2-yl]methyl}methanesulfonamide