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4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1,4-oxazepane
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-4,6-dimethylpyrimidin-2-amine
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]thiophene-3-carboxamide
ethyl 2-({2-[ethyl(oxan-4-ylmethyl)carbamoyl]phenyl}amino)acetate
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-fluorophenyl)urea
[(1-methyl-1H-indol-3-yl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
ethyl 3-{[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]amino}propanoate
N-({1-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)-3-hydroxypyridine-2-carboxamide
8-[3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(2-cyclooctyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)-N-(1-hydroxy-2-methylpropan-2-yl)piperidine-3-carboxamide
ethyl 5-({[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amino}methyl)-1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-1H-pyrazole-4-carboxylate
2-methoxy-1-[3-(3-methylphenoxymethyl)piperidin-1-yl]ethan-1-one
N-[2-(2-fluorophenyl)ethyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-3-phenoxy-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-(pyridin-3-ylmethyl)cyclopropanamine
1-(5-acetyl-2-ethoxyphenyl)-3-[2-(5-methylthiophen-2-yl)ethyl]urea
[2-(3,5-dimethyl-1H-pyrazol-4-yl)phenyl]methanol
(2R,6R)-4-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-6-carboxylic acid
2-(2-phenyl-1H-imidazol-1-yl)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}acetamide
N-[(3S,4R)-1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
dimethyl[2-({1-[(3-methyl-1-benzofuran-2-yl)methyl]piperidin-4-yl}oxy)ethyl]amine
3-(4-methylphenyl)-N-{2-[3-(1,2-oxazolidin-2-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}propanamide
1-(2-methoxyphenyl)-3-{1-[1-(4,4,4-trifluorobutanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-(2-fluorophenyl)-2-hydroxy-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}acetamide
N-(1-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
methyl 3-(cyclobutylmethoxy)-5-[methyl(piperidin-4-yl)carbamoyl]benzoate
9-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-butyl-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-[7-(1-benzothiophen-3-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
2-[2-ethoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
N-ethyl-6-[4-(3-fluorophenoxy)piperidin-1-yl]-N-methylpyridine-3-carboxamide
2-(ethylsulfanyl)-6-(4H-1,2,4-triazol-4-yl)-1,3-benzoxazole
4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-N-methylpyridin-2-amine
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-(9H-fluoren-9-yl)acetamide
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]amine
2-(azepan-1-yl)-2-[4-(3-hydroxypropyl)phenyl]acetic acid
4-{[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]sulfamoyl}-N-(2-hydroxyethyl)benzamide
2-ethyl-4-[(4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazin-1-yl)methyl]pyrimidine
(2E)-N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-(4-methoxyphenyl)prop-2-enamide
4-hydroxy-4-(hydroxymethyl)-N-(naphthalen-1-yl)azepane-1-carboxamide
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-N-[(4-fluorophenyl)methyl]propanamide
2-methoxy-4-methyl-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)benzene-1-sulfonamide
2-amino-6-(1H-indol-3-yl)-4-(pyridin-4-yl)pyridine-3-carbonitrile
2-methyl-1-[4-(4-methylphenoxy)piperidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
3-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(ethylamino)pyrimidine-5-carboxamide
7-(2,2-dimethylpropyl)-2-(5-methyl-1H-indazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
3-(2,6,8-trimethylquinoline-4-amido)pyrrolidine-3-carboxylic acid
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl)[2-(morpholin-4-yl)propyl]amine