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N-(3-phenylprop-2-yn-1-yl)-N-propylimidazo[1,2-a]pyridine-3-carboxamide
6-fluoro-2-oxo-N-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
(1R,6S)-3-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)-9-methyl-3,9-diazabicyclo[4.2.1]nonane
N-(1-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N,2-dimethylfuran-3-carboxamide
1-(2-methoxyethyl)-6-oxo-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidine-3-carboxamide
8-chloro-2-(furan-2-yl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]quinoline-4-carboxamide
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-2-[(4-hydroxyquinazolin-2-yl)sulfanyl]acetamide
9-[(5-chlorothiophen-2-yl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-N,N-dimethylaniline
1,3-dimethyl-6-[(1S,5R)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(1H-indol-4-ylmethyl)-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
N-[(2,5-dimethylphenyl)methyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
(4aS,7aR)-1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(4-cyanophenyl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(morpholin-4-yl)ethan-1-one
N-(3-chloro-4-fluorophenyl)-3-{1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}propanamide
6-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purine
N-[5-({[2-(cyclohexylsulfanyl)ethyl]carbamoyl}amino)-2-methoxyphenyl]acetamide
3-cyclopropyl-N-methyl-N-(quinolin-5-ylmethyl)-1,2-oxazole-5-carboxamide
2-(4-methylpiperazine-1-carbonyl)-6-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyrazine
4-(4-{[(2,6-difluoro-3-methylphenyl)methyl]amino}piperidin-1-yl)-N,N-dimethylbenzamide
5-cyano-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N,2,5-trimethyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-methoxyacetamide
3-[(4-methoxyphenyl)methyl]-1-methyl-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[(methylsulfanyl)methyl]-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-4-[2-(thiophen-3-yl)acetyl]-1,4-diazepan-2-one
3-(dimethyl-1,2-oxazol-4-yl)-N-[(4-methanesulfonylmorpholin-2-yl)methyl]propanamide
(furan-2-ylmethyl)(prop-2-en-1-yl){[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}amine
(3S,7S,8aS)-3-(1H-indol-3-ylmethyl)-7-{[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-(2-methylbutan-2-yl)acetamide
(4aR,7aS)-1-(2-methylpropanoyl)-4-(1H-pyrazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{4-[5-(furan-3-yl)-1,2,4-oxadiazol-3-yl]phenyl}ethan-1-ol
2-({4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)-1,3-benzothiazole
2-[(6-methyl-2-propylpyrimidin-4-yl)amino]-N-(1,3-thiazol-2-yl)acetamide
(2-{1-[(2-cyclohexylpyrimidin-5-yl)methyl]piperidin-2-yl}ethyl)dimethylamine
1-{2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-4-(thian-4-yl)piperazine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(5-chlorothiophene-2-carbonyl)pyrrolidin-3-yl]methanol
2-(2-methoxyethyl)-8-[2-(pyridin-4-ylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-(2H-1,3-benzodioxole-5-carbonyl)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(methylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
methyl 1-[(3S,5S)-1-(thiophen-3-ylmethyl)-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
5-{1-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-imidazol-2-yl}-2-(thiophen-2-yl)pyrimidine
3-[1-(3-methoxybenzoyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-(quinoxaline-5-carbonyl)piperidin-4-ol
(3R,4S)-1-[(4-methylthiophen-2-yl)sulfonyl]-4-propylpyrrolidin-3-amine
1-(morpholin-4-yl)-2-[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-methoxy-1-(2-{1-methyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one