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4-[1-(furan-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-3-phenyl-1H-pyrazole
1-(ethanesulfonyl)-3-[2-(2-fluorophenyl)ethyl]piperidine
3-{2-[3-(2-methylphenoxy)azetidin-1-yl]-2-oxoethyl}-4-(propan-2-yl)piperazin-2-one
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-(4-fluoro-2-methylphenyl)-3-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
N-cyclopentyl-2-fluoro-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}benzamide
1-[1-(hydroxymethyl)-9-[(3-methylpyrazin-2-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-(methylsulfanyl)ethan-1-one
2-{2-[1-(1H-indole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
(2S,4R)-4-amino-N-ethyl-1-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]pyrrolidine-2-carboxamide
3-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-1-(4-ethylpiperazin-1-yl)propan-1-one
3-{[3-(aminomethyl)pyrrolidin-1-yl]methyl}-2,4-dichlorophenol
1-(2-{[4-(cyclopropylmethyl)piperazin-1-yl]methyl}-5-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
(3S,7S,8aS)-7-(benzylamino)-3-methyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-ethyl-N-(oxan-4-ylmethyl)piperidin-3-amine
(1S,5R)-3-methyl-6-[(2,3,4-trimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
2-[(3-methoxyphenyl)methyl]-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[4.5]decan-3-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]propan-1-one
ethyl 4-oxo-5-phenoxy-1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1,4-dihydropyridine-3-carboxylate
5-cyclopropyl-N-[2-(diethylamino)ethyl]-N-ethyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
[(3S,4S)-4-(hydroxymethyl)-1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methanol
4-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
3-(2-ethyl-1H-1,3-benzodiazol-6-yl)-1-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]urea
1-(cyclohexylmethyl)-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine
2-methoxyethyl (3S)-3-(tert-butylcarbamoyl)-1,2,3,4-tetrahydroisoquinoline-2-carboxylate
2-{4-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-1,4-diazepan-1-yl}-4,6,7-trimethylquinazoline
3-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)sulfonyl]-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-methylpiperazine-1-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)pyrazine-2-carboxamide
4-(4-{[3-(2-hydroxyethyl)-4-[(2-methylphenyl)methyl]piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
5-(diethylamino)-1-methyl-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
propan-2-yl 4-{3-[(2-phenylethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxylate
2-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-N,N-dimethylaniline
4-(1,3-benzothiazol-2-yl)-2-(morpholin-4-ylmethyl)phenol
1-{3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
8-(2-amino-6-methoxypyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
2-amino-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-4-methyl-1,3-benzothiazole-6-carboxamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]piperidin-3-yl]methanol
3,4,7-trimethyl-2-[3-(morpholin-4-yl)azetidine-1-carbonyl]-1H-indole
5-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-methyl-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-5-(4-methylpent-3-en-1-yl)piperidin-2-one
2,8-dimethyl-N-(2-methylbut-3-yn-2-yl)quinoline-4-carboxamide
2-[1-(3-phenylpropyl)-4-(quinolin-4-yl)piperazin-2-yl]ethan-1-ol
2-[2-(4-fluorophenyl)ethyl]-4-[4-(2-methoxyacetyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-{4-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]piperazin-1-yl}pyridine-3-carboxamide
4-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
2-[(4-acetamidopiperidin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid