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4-ethyl-1-methyl-3-{1-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-5-methyl-1,2-oxazole-4-sulfonamide
1-ethyl-5-(4-phenyl-1H-imidazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-{4-[(5-ethylpyridin-2-yl)methyl]-2-oxopiperazin-1-yl}benzonitrile
N-methyl-2-(methylamino)-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}pyridine-4-carboxamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2-methylbenzamide
N-methyl-6-(piperidin-1-yl)-N-(1,3-thiazol-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-(1,4-dioxan-2-ylmethyl)-6-{[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
{[5-(4-chloro-2-fluorophenyl)furan-2-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
5-methyl-6-(4-methylpiperidine-1-carbonyl)-N-(pyridin-2-ylmethyl)thieno[2,3-d]pyrimidin-4-amine
1-{2,7-diazaspiro[4.5]decan-7-yl}-2-methyl-2-(1H-pyrrol-1-yl)propan-1-one
N-[4-(N-methylacetamido)phenyl]-2-{[2-(thiophen-2-yl)ethyl]amino}acetamide
7-(cyclopropylmethyl)-2-[(1-propyl-1H-pyrazol-5-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4-fluorophenyl)ethyl]-5-{4-hydroxy-1-[(4-methylphenyl)methyl]piperidin-4-yl}-1-benzofuran-2-carboxamide
N-[(2,2-dimethyloxan-4-yl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
2-(5-methyl-1,2-oxazol-3-yl)-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidine
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]cyclobutanecarboxamide
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-2-(oxan-2-ylmethoxy)acetamide
3-hydroxy-1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-(3-hydroxyphenyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
4-methyl-2-{[2-(1-phenylethyl)-1H-imidazol-1-yl]methyl}-1,3-thiazole
8-fluoro-3-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]-1,4-dihydroquinolin-4-one
N,N-diethyl-2-[4-ethyl-5-oxo-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
N-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
[(3-fluorophenyl)methyl]({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})amine
6-[(3S,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
5-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-2-methoxybenzamide
[(dimethyl-1,2-oxazol-4-yl)methyl]({[3-(ethoxymethyl)-4-methoxyphenyl]methyl})methylamine
2-[1-(5-chlorothiophene-2-carbonyl)pyrrolidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-3-(morpholin-4-yl)propanamide
methyl(oxolan-3-ylmethyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methylpiperazine
2-methoxyethyl 8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxylate
3-(dimethyl-1,2-oxazol-4-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]propan-1-one
2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-1-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}piperidine
4-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-2,6-dimethylpyridine
(3R,4S)-1-(2-chloro-6-methylbenzenesulfonyl)-4-cyclopropylpyrrolidin-3-amine
methyl 6-(2-cyclopropylacetyl)-2-{[(3,4-difluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N,N-dimethyl-2-(pyridin-4-yl)-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(cyclopropylmethyl)-N-methyl-5-[2-(pyridin-3-yl)acetyl]-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1R,5R)-6-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-methyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]imidazo[1,2-a]pyrimidine-3-carboxamide
3-chloro-4-({1-[(3-fluorophenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
2,6-diamino-4-[4-(1H-pyrazol-1-yl)phenyl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
2-{[2-(4-chloro-3-methyl-1H-pyrazol-1-yl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
4-{5-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-1H-pyrazol-3-yl}phenol
4,4,4-trifluoro-1-[3-(2-phenylacetyl)piperidin-1-yl]butan-1-one