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2-(3-{[4-(2-methoxyphenoxy)piperidin-1-yl]methyl}phenoxy)acetamide
ethyl 4-[3-(4-methylphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperazine-1-carboxylate
2-butyl-8-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(2,6-dimethylpyridin-4-yl)-4-(3-phenyl-1,2-oxazole-4-carbonyl)piperazine
N-{4-[2-(dimethylamino)ethoxy]-1-(3-fluorophenyl)-1H-indazol-3-yl}-1,2-oxazole-3-carboxamide
4-[(1-cyclohexyl-3-methyl-1H-1,2,4-triazol-5-yl)(pyridin-3-yl)methyl]morpholine
N4,5-dimethyl-N4-(quinolin-8-ylmethyl)pyrimidine-2,4-diamine
5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
1-(2,6-difluoro-3-methoxybenzoyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N-methyl-2-oxo-N-[1-(3-phenylpropyl)piperidin-3-yl]-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
3-(4-fluorophenyl)-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazin-2-one
6-methoxy-1-[(4-methoxyphenyl)methyl]-4-(1H-pyrazol-3-ylmethyl)-1,4-diazepan-2-one
4-{[4-methyl-5-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}morpholine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}acetamide
1-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)urea
1-(2-methoxyethyl)-4-oxo-N3-[(1-phenylcyclopentyl)methyl]-N5-[2-(propan-2-yloxy)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-4-(1H-imidazol-1-yl)-N-(2-methoxyethyl)benzamide
2-(methylsulfanyl)-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
2-amino-2-methyl-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)propan-1-one
N-[3-(4-{[3-(1H-1,2,3-benzotriazol-1-yl)propyl]amino}piperidin-1-yl)phenyl]-2-methoxybenzamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
ethyl 3-benzyl-1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidine-3-carboxylate
2-methoxy-5-{1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}benzoic acid
ethyl 5-(1H-imidazol-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-butyl-1'-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N6-cyclopentyl-N5-methyl-N5-[2-(morpholin-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-S-(4-fluoro-2-methylphenyl)-2-oxoethane-1-sulfonamido
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1,3-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}-1,4-oxazepane
(3S,4S)-1-{[4-(benzyloxy)phenyl]methyl}-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
6-oxo-4-(2-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylic acid
2-(1H-1,3-benzodiazol-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
3-({2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}sulfonyl)benzonitrile
3-{2-[4-(4-acetylphenyl)piperazin-1-yl]-2-oxoethyl}-4-(2-methylpropyl)piperazin-2-one
N-ethyl-2-(5-methoxy-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-(2-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[(4aR,7aS)-6,6-dioxo-4-(propane-1-sulfonyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
methyl[(3-methylthiophen-2-yl)methyl][1-(pyrazin-2-yl)propan-2-yl]amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-ethyl-N,4-dimethyl-1,3-thiazole-5-carboxamide
3-(2-methoxyphenyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-5-carboxamide
3-({1-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)morpholine
5-fluoro-2-(1-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
1-(3-chlorophenyl)-4-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}piperazin-2-one
methyl({[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}){[3-(trifluoromethyl)phenyl]methyl}amine
3-(1-methyl-1H-pyrazol-4-yl)-1-{1-oxa-8-azaspiro[4.6]undecan-8-yl}propan-1-one
3-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}pyridin-2-ol
N-[4-(2,2-dimethylpropanamido)-3-methylphenyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
5-[({[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]pyrimidin-2-amine
2-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-4-methylphenol