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2,5-dimethyl-1-phenyl-N-[(2R)-pyrrolidin-2-ylmethyl]-1H-pyrrole-3-carboxamide
1-{1-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]piperidin-4-yl}piperidin-3-ol
(2E)-3-(2-chlorophenyl)-N-{[4-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)prop-2-enamide
1-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}azetidin-3-ol
N,N-dimethyl-1-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-amine
1-{[(2-methoxy-5-methylphenyl)carbamoyl]methyl}-5-oxopyrrolidine-3-carboxylic acid
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(2,1,3-benzothiadiazol-5-ylmethyl)methylamine
2-[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]pyridine-3-carboxylic acid
N-[2-(4-cyclohexylmorpholin-2-yl)ethyl]-2-(2-oxopyrrolidin-1-yl)acetamide
N-(2,2-dimethyloxan-4-yl)-N-ethyl-4-hydroxy-2-methylpyrimidine-5-carboxamide
8-fluoro-3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-1,4-dihydroquinolin-4-one
N-cyclohexyl-3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)propanamide
1-(2-chlorophenyl)-3-(1-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-(1,2-oxazol-3-ylmethyl)benzamide
2-{[4-(2-amino-6-methylpyrimidin-4-yl)piperazin-1-yl]methyl}benzoic acid
[(3R,5R)-5-[(dimethylamino)methyl]-1-[2-(4-fluorophenyl)benzoyl]piperidin-3-yl]methanol
1-ethyl-N-[2-(5-methylfuran-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
3-[3-(2-oxopyrrolidin-1-yl)propyl]-1-(3-phenylphenyl)urea
(4aS,7aR)-1-(1H-indole-2-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-chlorophenyl)-3-methyl-N-(2-propoxyethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-phenoxy-1-(4,4,4-trifluorobutanoyl)piperidine-4-carboxylic acid
1-(2,1,3-benzoxadiazol-5-ylmethyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
N-[2-(4-fluorophenyl)ethyl]-3-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1,2-oxazole-5-carboxamide
2-methyl-3-(2-{[6-(piperidin-3-yl)pyrimidin-4-yl]amino}ethyl)-1H-indole-5-carbonitrile
1-(diethylamino)-3-[2-methoxy-4-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-methyl-2-(3-phenylpyrrolidin-1-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[2-(4-methylpentyl)morpholin-4-yl]propan-1-one
N-[2-(azepan-1-yl)-2-phenylethyl]-3-methyl-1,2-oxazole-5-carboxamide
3-{[(5-methyl-1,2-oxazol-3-yl)methyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-{2-[(3-methoxyphenyl)methyl]morpholine-4-carbonyl}benzonitrile
(1R,5S)-3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-methoxyethan-1-one
3-ethyl-5-methyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,2-oxazole
4-(4-{1-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}phenyl)-2-methylbut-3-yn-2-ol
2-methoxy-N,N-dimethyl-5-({[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]carbamoyl}amino)benzamide
1-{4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecan-11-yl}-2-methylpropan-1-one
4-[(E)-2-phenylethenesulfonyl]piperazine-2-carboxylic acid
4-{6-[5-chloro-2-(propan-2-yloxy)phenyl]pyridine-3-carbonyl}morpholine
7-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
8-chloro-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylquinoline-2-carboxamide
2-[(2-{[2-(dimethylamino)-6-methylpyrimidin-4-yl]oxy}hex-5-en-1-yl)(methyl)amino]-N,N-dimethylacetamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-4-(thiophen-2-yl)butanamide
N-methyl-N-[2-(oxan-2-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
2-({3-[2-(3-hydroxyphenyl)pyridin-4-yl]pyrrolidin-1-yl}methyl)-6-methoxyphenol
3-{2-[1-(2,5-difluorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyridine
2-(naphthalen-2-yloxy)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(pyridazine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-({1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
2-(3-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}piperidin-1-yl)acetamide