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N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(2-oxopyrrolidin-1-yl)propanamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-[1-(pyridin-4-yl)propyl]-1,2-oxazole-3-carboxamide
2-cyclopropyl-9-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-2-(2,4-difluorophenoxy)-N-(thiophen-3-ylmethyl)acetamide
5-{4-[1-(dimethylamino)ethyl]phenyl}pyridin-2-amine
1-methyl-6-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}-1H-indole
ethyl 3-[(3-chlorophenyl)methyl]-1-(3-methoxypropanoyl)piperidine-3-carboxylate
4-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazole
2-[2-(dimethyl-1,3-thiazol-5-yl)-N-methylacetamido]-N-methylpropanamide
3-(prop-2-en-1-yl)-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}piperidine-3-carboxylic acid
N-benzyl-N-methyl-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-3-amine
3-(dimethyl-1,2-oxazol-4-yl)-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]propanamide
1-(2,4-difluorobenzoyl)-3-ethylpiperidine-3-carboxylic acid
8-(4-cyclopropanecarbonyl-3-fluorophenyl)quinoline
1-(1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)pyrrolidin-2-one
1-{pyrazolo[1,5-a]pyridine-3-carbonyl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
3-(5-chlorothiophen-2-yl)-5-methoxypyridine
1-(3-ethyl-1H-pyrazole-5-carbonyl)-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(1S,5R)-3-(oxan-4-yl)-6-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
5-{1-[1-(5-methylpyridin-2-yl)ethyl]-1H-imidazol-2-yl}-2-(thiophen-2-yl)pyrimidine
8-(6-aminopyridine-3-carbonyl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1,3-dimethyl-N-[(1-methylpiperidin-2-yl)methyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-ethyl-2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}acetamide
4-(2-fluorophenoxy)-1-(oxolan-3-ylmethyl)piperidine-4-carboxylic acid
3-(4-{2-amino-6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}phenyl)propanoic acid
N-[(2-amino-1,3-thiazol-4-yl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
4-({1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]piperidin-2-yl}methyl)morpholine
1,5-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-pyrrole-2-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-[methyl(2-phenylethyl)amino]piperidine-1-carboxamide
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(5-methylfuran-2-yl)methyl]-3-{1-[3-(thiophen-3-yl)propanoyl]piperidin-3-yl}propanamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{3-[5-(1,2-oxazol-3-yl)thiophen-2-yl]phenyl}acetamide
1-(morpholin-4-yl)-2-[4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazin-1-yl]ethan-1-one
methyl 2-[methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]acetate
N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetamide
(3S,9aR)-8-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-2,3-dimethyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-3-phenylpropan-1-ol
3-[1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-yl]-1,3-oxazolidin-2-one
methyl 5-(3-hydroxypropanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1,7-dimethyl-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
2-(4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
4-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]azetidin-3-yl}morpholine
1-(furan-2-ylmethyl)-N-[(2-propyl-1,3-thiazol-4-yl)methyl]piperidine-3-carboxamide
(1S,5R)-6-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-methoxyethyl)-3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{1-[(5-methylpyrazin-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
2-(2-ethoxypyridin-3-yl)-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]acetic acid
[3-(cyclopropylmethyl)-1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-3-yl]methanol
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide