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5-[1-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-3-yl]-4-methyl-N-(thiophen-2-ylmethyl)-1,3-thiazol-2-amine
N-[(3S,4R)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-{1-[1-(1-benzofuran-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
4-[(5-chlorothiophen-2-yl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
(benzylsulfamoyl)(methyl)[3-(oxolan-2-yl)propyl]amine
2-(1,3-thiazol-4-yl)-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
3-butyl-4-(4-methoxyphenyl)-4H-1,2,4-triazole
6-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine-4-carbonyl}-2-methyl-1,3-benzothiazole
4-[4-(1H-pyrazol-3-yl)benzamido]oxane-4-carboxylic acid
[3-(1H-imidazol-4-ylmethyl)-9-(pyridin-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
3-{[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]methyl}benzonitrile
(3-{2-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}phenyl)methanol
1-[4-(3-{[(naphthalen-1-ylmethyl)amino]methyl}pyridin-2-yl)piperazin-1-yl]ethan-1-one
N-[(3S,4R)-4-(4-methylphenyl)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-3-yl]acetamide
1-{2-[4-(2-methoxyethoxy)phenyl]pyrimidin-4-yl}piperidin-4-ol
2-(2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydroisoquinolin-1-one
(2S,4S)-4-{[(9-ethyl-9H-carbazol-3-yl)methyl]amino}-1-(naphthalen-1-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-2-(2-hydroxyphenoxy)ethan-1-one
2-(8-methylquinolin-5-yl)benzamide
3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
4-[4-(4-methylphenoxy)piperidin-1-yl]-6-(morpholin-4-yl)pyrimidin-2-amine
1-(5-hydroxypyrazine-2-carbonyl)-4-(4-methylphenoxy)piperidine-4-carboxylic acid
1-(furan-2-ylmethyl)-4-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}piperidine
1-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)ethan-1-ol
[3-(5-chloro-2-ethoxyphenyl)-1H-1,2,4-triazol-5-yl]methanol
methyl 8-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
4-{[4-(benzyloxy)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
1-ethyl-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-methyl-N-[4-(pyridin-2-yl)butyl]-1-benzofuran-5-carboxamide
{9-[(2-ethylpyrimidin-5-yl)methyl]-3-(1H-imidazol-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
N-(2,2-dimethylpropyl)-N-ethyl-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
2-(3-methyl-1,2-oxazol-5-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1H-1,2,3-triazole
4-[3-(morpholin-4-ylmethyl)phenyl]-5H,6H,7H-cyclopenta[d]pyrimidin-2-amine
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methylimidazo[1,2-a]pyridine
2-{[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]methyl}quinolin-4-ol
3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]quinoline
N-[(3-methoxyphenyl)methyl]-4-methyl-5-{1-[2-(thiophen-2-yl)ethyl]-1H-pyrazol-3-yl}-1,3-thiazol-2-amine
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(2-methyl-1H-indol-3-yl)ethan-1-one
(2S,4S)-4-amino-N,N-diethyl-1-[(1s,4s)-4-hydroxycyclohexanecarbonyl]pyrrolidine-2-carboxamide
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-(morpholin-3-yl)ethan-1-one
(5S,9aS,9bS)-5-[4-(2-hydroxyethoxy)phenyl]-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(5-tert-butyl-2-methoxyphenyl)-3-methyl-3-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}urea
4-methoxy-N-methyl-3-({[2-methyl-1-(morpholin-4-yl)propan-2-yl]carbamoyl}amino)benzamide
2-{4-[(3,4-difluorophenyl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
(3aR,6aR)-2-methanesulfonyl-N-[2-(thiophen-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-(2-methyl-1,3-thiazole-4-carbonyl)-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
4-ethyl-2-methyl-5-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,3-thiazole