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methyl 5-(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
2-amino-2-methyl-1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]propan-1-one
4-cyclopropyl-5-[(5-propylfuran-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
N-({4-hydroxy-1-[2-(morpholin-4-yl)-2-oxoethyl]azepan-4-yl}methyl)benzamide
1-(1-methylcyclopropanecarbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
methyl 1-(naphthalen-2-ylmethoxy)-2-oxo-8-(pyridin-2-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-[(3-methoxyphenyl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
5-cyclobutanecarbonyl-1'-(5-methyl-1,3-oxazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-({1-[(5-methylthiophen-2-yl)sulfonyl]piperidin-3-yl}methyl)furan-2-carboxamide
7-cyclohexyl-2-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
5-[(4-acetyl-4-phenylpiperidin-1-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}propanamide
methyl (2S)-3-(1H-indol-3-yl)-2-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}propanoate
N-benzyl-N-methyl-3-[1-(3-phenoxypropanoyl)piperidin-4-yl]propanamide
2-(2-chlorophenyl)-3-methyl-N-(4,4,4-trifluorobutyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(4-{2-[(2,4-dimethoxyphenyl)carbamoyl]acetyl}morpholin-3-yl)acetic acid
3-(2H-1,3-benzodioxol-5-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
2-methyl-5-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
2-amino-8-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1-ethyl-N-[4-(furan-2-yl)butan-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
N-[(3S,4R)-4-(propan-2-yl)-1-(pyrimidin-5-ylmethyl)pyrrolidin-3-yl]methanesulfonamide
2-(5-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
2-[4-(hydroxymethyl)phenyl]-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethan-1-one
2-(2-hydroxypropanoyl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-oxo-2-phenylacetamide
4-(1-methyl-1H-imidazol-2-yl)-1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidine
2-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-4-methylphenol
2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
5-{2-[3-(dimethylamino)pyrrolidin-1-yl]pyrimidin-4-yl}-2-ethoxybenzoic acid
2-(2-fluoro-4-methylphenyl)-2-[4-(piperidine-1-carbonyl)piperidin-1-yl]acetic acid
1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]piperidin-4-amine
2-(adamantan-1-yl)-N-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]acetamide
5-{5-[2-(2-methoxyphenoxy)propan-2-yl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[3-(methylsulfamoyl)phenyl]-4-(oxan-4-yl)piperazine-1-carboxamide
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-1,1-dioxo-1λ6-thiane-4-carboxamide
1-cyclobutanecarbonyl-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,4-diazepane
(2R,3S,6R)-5-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[3-(3-chlorophenyl)phenyl]-1-[(4-hydroxyphenyl)methyl]piperidine-4-carboxamide
propan-2-yl 2-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxylate
{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
N-[2-(2,3-dimethoxyphenyl)ethyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-cyclopropyl-2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridine-4-carboxamide
4-(3,5-dimethoxyphenyl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[1-(furan-2-yl)ethyl]-N-methyl-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide