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2-amino-4-[2-(2-hydroxyethoxy)phenyl]-5-methyl-6-phenylpyridine-3-carbonitrile
1-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,3-benzodiazole
ethyl 4-[1-(1,2-oxazol-3-ylmethyl)piperidin-3-yl]piperazine-1-carboxylate
2-{1-[(2-fluoro-5-methoxyphenyl)methyl]pyrrolidin-2-yl}ethan-1-ol
(1R,7S)-N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-[2-(3-methoxypropyl)piperidine-1-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
1,1-dioxo-N-(5,6,7,8-tetrahydronaphthalen-1-yl)-1λ6-thiomorpholine-4-carboxamide
8-(4-aminopyrimidin-2-yl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(2-hydroxyethyl)-8-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
5-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-2-methoxybenzoic acid
4-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-N-methylpyridin-2-amine
5-(cyclohexylmethyl)-7-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
3-methyl-1-[(3-methylphenyl)methyl]-5-(oxan-4-yl)-1H,4H-pyrazolo[3,4-d]imidazole
9-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{3-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
[(4-ethylphenyl)methyl]({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
{2-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-2-yl]ethyl}dimethylamine
ethyl({[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl})(2-methylprop-2-en-1-yl)amine
N-(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
N-(2-hydroxyethyl)-5-methoxy-1-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-indole-2-carboxamide
2-({[(8-methoxyquinolin-5-yl)methyl](methyl)amino}methyl)-N-(thiophen-2-ylmethyl)quinazolin-4-amine
1-(cyclopropanesulfonyl)-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-[(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)methyl]-2-methoxyphenol
[(6-chloroquinolin-2-yl)methyl][(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
N-[1-(furan-2-carbonyl)piperidin-3-yl]-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
2-(3-{1-cyclohexyl-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenoxy)ethan-1-ol
(4S,4aS,8aS)-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4-phenyl-decahydroquinolin-4-ol
4-{6-[3-(1H-pyrazol-3-yl)phenyl]pyridine-3-carbonyl}morpholine
1-(2-ethoxyethyl)-5-(5-oxo-1,4-diazepane-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-methyl-2-phenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-imidazole-4-carboxamide
6-(1-benzofuran-2-ylmethyl)-N-(3,4-difluorophenyl)-6-azaspiro[2.5]octane-1-carboxamide
7-[(4-methoxynaphthalen-1-yl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-(butan-2-yl)-5-[2-(difluoromethoxy)phenyl]-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
3-(1-methyl-1H-pyrazol-4-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-benzyl-9-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-1-(pyrrolidin-1-yl)propan-1-one
(2S,4R)-N-[2-(3-fluorophenyl)ethyl]-1-[(4-fluorophenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carboxamide
2-methyl-7-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-2,7-diazaspiro[4.4]nonane
1-methyl-4-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperazine-2-carboxylic acid
3-(2-methoxyethyl)-3H,4H-pyrido[4,3-d]pyrimidin-4-one
2-(2-oxopyrrolidin-1-yl)-N-[(3R,4S)-4-propyl-1-(pyrazin-2-yl)pyrrolidin-3-yl]acetamide
N-{[1-(3,5-dimethylfuran-2-carbonyl)piperidin-3-yl]methyl}-4-methoxybenzene-1-sulfonamide
3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)propanamide
N-{2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-oxoethyl}acetamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
2-{4-[(3-oxopiperazin-1-yl)methyl]phenyl}-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
[(2S,6S)-11-methoxy-4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
6-(1-benzofuran-3-carbonyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine