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2-(2H-1,3-benzodioxol-5-yl)-4,6-dimethylpyridine-3-carboxamide
N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
4-{7,11-dimethyl-3,7,11-triazaspiro[5.6]dodecane-3-carbonyl}pyridin-3-ol
(4aS,8aR)-6-(4-methylbenzenesulfonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
9-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
3-hydroxy-S-[3-(2-phenylazetidine-1-carbonyl)phenyl]propane-1-sulfonamido
1-[(4-fluorophenyl)methyl]-5-[3-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
2-[(1S,5R)-6-[5-(hydroxymethyl)furan-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[(oxan-4-ylmethyl)amino]pyridine-3-carboxamide
4-benzyl-1-{2-[4-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
2-(morpholin-4-yl)-2-(pyridin-3-yl)-1-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethan-1-one
1-[2-(3-fluorophenyl)ethyl]-5-[4-(6-methylpyridin-2-yl)piperazine-1-carbonyl]piperidin-2-one
methyl 6-(2-cyclopropylacetyl)-2-{[(3-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-{[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-1-phenylpyrrolidin-2-one
3-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}benzoic acid
5-benzyl-5-[1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-(3-methoxypropyl)-N-methylacetamide
3-methyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}butan-1-ol
2-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-N-(1,3-thiazol-2-yl)acetamide
2-(3-fluorophenoxymethyl)-1,3-oxazole-4-carboxylic acid
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-N-[(4-methoxyphenyl)methyl]piperidine-1-carboxamide
4-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}morpholine
1-(4-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-4-oxobutyl)pyrrolidin-2-one
(1S,5R)-3-(4-chloro-1H-indole-2-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-methyl-9-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4-phenyl-2,9-diazaspiro[5.5]undecane
1-cyclohexyl-3-(cyclopropylmethyl)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
7-fluoro-4-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1,2-dihydroquinolin-2-one
4-({5-[1-(2,6-dimethylpyridin-4-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
3-(2H-1,3-benzodioxol-5-yl)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}propanamide
(3aR,6aR)-N-{[1-(3-fluorophenyl)cyclopentyl]methyl}-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-2-(methoxymethyl)-6-methyl-1-(3-phenylpropyl)-1,4-dihydropyridin-4-one
4-(2,2-diphenylethyl)-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]piperazin-2-one
[1-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)cyclopropyl]methanol
2-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-2-yl)acetic acid
3-(2H-1,3-benzodioxol-5-yl)-1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}propan-1-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-N'-(2-methylphenyl)propanediamide
4-[(2,3-dichlorophenyl)methyl]-4H-1,2,4-triazole
4-{[1-(cyclopropylmethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}-1-[(4-methylphenyl)methyl]piperazin-2-one
(3S,4R)-4-(2-methylphenyl)-1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidine-3-carboxylic acid
N-[(4-methylphenyl)(pyridin-4-yl)methyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
3-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]-1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]urea
4-{[(3-fluorophenyl)methyl]amino}-5-methyl-N-[3-(morpholin-4-yl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
3-[1-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)azetidin-3-yl]pyridine
1-methyl-2-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1H-1,3-benzodiazole
2-methyl-4-[5-({3-[methyl(2-phenylethyl)amino]piperidin-1-yl}methyl)thiophen-2-yl]but-3-yn-2-ol
(5-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
{4-[(1-phenyl-1H-pyrazol-4-yl)methyl]morpholin-3-yl}methanol
4-chloro-1,3-dimethyl-N-[1-(thiophen-2-yl)propyl]-1H-pyrazole-5-carboxamide
(3S,4R)-1-(cyclopropanesulfonyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-methylpyridine