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ethyl({2-[4-(furan-2-ylmethyl)morpholin-2-yl]ethyl}sulfamoyl)methylamine
N-[2-(4-fluorophenyl)ethyl]-2-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}acetamide
4-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}piperazin-2-one
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
(3S,4S)-1-(benzenesulfonyl)-4-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}pyrrolidin-3-ol
3-chloro-4-[4-(dimethylcarbamoyl)phenyl]benzoic acid
2-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}-N-(2,3,4-trifluorophenyl)acetamide
N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}cyclohexanecarboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-(1H-pyrazol-1-yl)butanamide
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]propan-1-one
N-[3-(methylsulfanyl)propyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
2-[({5-[1-(4,6-dimethylpyrimidin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-phenylpiperidine-4-carbonitrile
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(thiophene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]pyrazine-2-carbonitrile
1-{4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-{4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidine
N-{2-[(E)-2-(8-hydroxyquinolin-2-yl)ethenyl]phenyl}-1H-pyrazole-3-carboxamide
N-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-4-(4-methyl-1H-pyrazol-3-yl)piperidine-1-carboxamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[2-(1H-pyrazol-1-yl)ethyl]amine
1-[(5-methylfuran-2-yl)methyl]-4-oxo-5-(3-oxo-4-phenylpiperazine-1-carbonyl)-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
7-methyl-3-[(8-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
(1S,5R)-3-(2,3-dimethyl-1H-indole-5-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
cyclopentyl 4-(3-acetamidobutanamido)benzoate
1-(2,4-difluorophenyl)-5-[1-(1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazole
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-(4-methylphenyl)-N-(oxolan-2-ylmethyl)propanamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(propan-2-yl)carbamoyl]-1,4-diazepane-6-carboxylic acid
methyl 4-({3-[(pyridin-2-ylformamido)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)benzoate
N-[3-(3-chlorophenyl)phenyl]-1-[(2-propylpyrimidin-5-yl)methyl]piperidine-4-carboxamide
4-(2-{[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]amino}ethyl)phenol
3-[1-(5-acetylthiophene-2-carbonyl)piperidin-3-yl]-N-[(2-chlorophenyl)methyl]propanamide
1-{3-[3-(2-chlorophenoxy)azetidin-1-yl]-3-oxopropyl}azepan-2-one
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
2-(5-acetylthiophen-3-yl)-1-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-[2-(4-fluorophenyl)ethyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-[2-(methylsulfanyl)ethyl]acetamide
(3S,4S)-4-(naphthalen-2-yl)-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-ol
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-(thiophen-2-yl)butan-1-one
2-(4-hydroxyphenyl)-7-(3-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(oxolane-2-carbonyl)-1,4-diazepane
(2S,4S)-4-amino-N-ethyl-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]pyrrolidine-2-carboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl]propanoic acid
N-[3-methoxy-4-(3-methylbutanamido)phenyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
(2-{[(6-methoxypyridin-3-yl)methyl](thiophen-3-ylmethyl)amino}ethyl)dimethylamine
1-benzyl-N,N-dimethyl-5-{methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[(2S)-1-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]pyrrolidine-2-carbonyl]morpholine
N-[1-(4-methanesulfonylphenyl)propyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-butyl-3-cyclopropyl-5-[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]-1H-1,2,4-triazole