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N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
9-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-3,9-diazaspiro[5.6]dodecane
5-(3-methoxyphenyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2,4-triazin-3-amine
1-(1-ethyl-1H-pyrazole-3-carbonyl)-4-(2-methoxyphenoxy)piperidine
methyl 3-(oxolane-3-amido)-1-(2-phenylethyl)-5-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)azetidin-3-yl]pyridine
4-(3-hydroxyphenyl)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)piperazine-1-carboxamide
2-[(3-chlorophenyl)methyl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide
(3S,4R)-1-(3-methanesulfonylpropanoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-methyl-1H-imidazole-2-carboxamide
N-(pyridin-3-yl)-2-[2-(pyrrolidin-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-[(7-{[5-(methoxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine-2-carboxamide
{1-[4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]piperidin-4-yl}(thiophen-2-yl)methanol
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-3-(thiophen-2-yl)propan-1-one
4-{2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}-1-phenylpiperazin-2-one
1-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyridin-2-ylmethyl)acetamide
9-(1H-pyrazole-4-sulfonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-cyclopropyl-6-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidine
propan-2-yl 3-{[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]amino}-4-chlorobenzoate
N-[1-(1,1-dioxo-1λ6-thian-4-yl)piperidin-4-yl]-1-methyl-1H-indole-6-carboxamide
2-(4-{[4-(cyclopentyloxy)phenyl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-(2-{4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}propyl)phenol
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N,2-dimethylimidazo[1,2-a]pyridine-6-carboxamide
N4-methyl-N4-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
5-{[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-4-methyl-1H-imidazole
4-phenyl-3-{1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2-chloro-4-fluorophenyl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
(1R,5R)-N,N-dimethyl-6-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
methyl 3-[(3S,4R)-4-(dimethylamino)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]propanoate
1-(azocan-1-yl)-3-(5-methoxy-2-{[(2-methoxyethyl)(methyl)amino]methyl}phenoxy)propan-2-ol
3-(1H-pyrazol-1-ylmethyl)-N-[1-(thiophen-2-yl)propan-2-yl]benzamide
N-[2-(azepan-1-yl)ethyl]-N-ethyl-1-propyl-1H-pyrazole-5-carboxamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-5,6-dimethylthieno[2,3-d]pyrimidine
8-(trimethyl-1H-pyrazole-4-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
methyl 4-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)benzoate
N-{1-[1-(2,2-difluoroethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
N-(5-chloro-2-methoxyphenyl)-3-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)propanamide
3-[(3R,4S)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(dimethylamino)piperidin-3-yl]propanoic acid
1-(3-methoxyphenyl)-4-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperazin-2-one
2-{4-[3-(cyclopropylcarbamoyl)piperidin-1-yl]piperidin-1-yl}acetic acid
N-methyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl 3-(2-chlorobenzenesulfonamido)-5-[(pyridin-2-ylformamido)methyl]benzoate
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-1,3-thiazole-5-carboxamide
3-methyl-7-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-phenylcyclopropane-1-carboxamide
methyl 2-{2-[6-(dimethylcarbamoyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-yl]acetamido}acetate