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6-[3,5-bis(trifluoromethyl)benzoyl]-2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-(carbamoylmethyl)-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]piperidine-4-carboxamide
N-[2-(4-methylbenzenesulfonyl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-[3-(4-cyano-4-phenylpiperidine-1-carbonyl)piperidin-1-yl]acetamide
N-[1-(1-{[5-(3-chlorophenyl)furan-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
3-chloro-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
4-{[1-(pent-4-enoyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
N-(2-methoxyethyl)-5-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrazine-2-carboxamide
3-{1-[3-(1H-indol-3-yl)propanoyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
3-[(1-butyl-3-methyl-1H-1,2,4-triazol-5-yl)methyl]-1H-indole
7-(2-phenylethyl)-2-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
4-[1-(propan-2-yl)piperidin-4-yl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-cyclopentyl-N-[2-(2,4-dimethoxyphenyl)ethyl]-5-oxopyrrolidine-3-carboxamide
1-[(2E)-3-phenylprop-2-en-1-yl]-4-(piperidine-1-sulfonyl)-1,4-diazepane
1-methyl-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-(1-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-2,3-dimethoxybenzamide
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
5,6-dimethyl-3-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydropyridin-2-one
1-[(9-ethyl-9H-carbazol-3-yl)methyl]-4-(2-methoxyethyl)-1,4-diazepan-5-one
N-benzyl({2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}amino)sulfonamide
7-(1-ethyl-3,5-dimethyl-1H-pyrazole-4-carbonyl)-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
12-(oxolan-2-ylmethyl)-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
2-ethyl-9-(5-methyl-1,2-oxazole-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
5-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)thiophene-2-carboxamide
2-(thiophen-3-ylmethyl)-4-(4-{[4-(trifluoromethoxy)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[1-(furan-2-carbonyl)piperidin-3-yl]-2,3,6-trimethylquinoline-4-carboxamide
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
2-[1-({1-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(5-ethyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-yl]methanol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-3-ol
{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}bis(1,3-oxazol-4-ylmethyl)amine
4-[2-(1-methylpiperidin-2-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
[2-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-2-oxoethyl]urea
1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-2-methyl-4-phenylpiperazine
N-[2-hydroxy-2-(1-methyl-1H-imidazol-2-yl)ethyl]-4-(4-methoxyphenoxy)benzamide
2-methyl-N-(1-phenylbutyl)furan-3-carboxamide
3-(4-methylphenyl)-1-[2-(morpholin-4-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
8-benzyl-3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(furan-2-yl)-1-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]azepane
1-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-3-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)urea
(1R,2S,4R)-N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
3-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-1-methyl-1-[1-(4-methylpyridin-2-yl)propan-2-yl]urea
N-benzyl-1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-4-carboxamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1,7-dimethyl-1H-indole-2-carboxamide
N2-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidine-2,4-diamine
2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]acetamide
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
8-[2-(2-hydroxyethoxy)ethyl]-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
(5-{[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}furan-2-yl)methanol
(3aS,6aS)-2-benzyl-5-(1H-imidazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid