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8-(morpholine-4-carbonyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(1-ethyl-1H-pyrazole-5-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2,3-dimethyl-6-{2-methylthieno[3,2-d]pyrimidin-4-yl}-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
9-(1-methylpiperidine-2-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-7-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-5-phenylpyrazolo[1,5-a]pyrimidine
4-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}-1-(2-methylbutyl)piperidine
3-(pyridin-2-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
dimethyl(3-{2-[1-(quinoline-7-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
N-[(3R,4S)-4-cyclopropyl-1-(2-methanesulfonylethyl)pyrrolidin-3-yl]-1,5-dimethyl-1H-pyrazole-4-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2,4-difluoro-3-methoxybenzamide
6-(cyclopropylmethoxy)-4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
(1R,2S,9R)-11-[(2-methyl-1,3-thiazol-4-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
[5-(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
ethyl 2,4-dimethyl-5-{[1-(2-phenylethyl)piperidin-3-yl]carbamoyl}-1H-pyrrole-3-carboxylate
3-(hydroxymethyl)-1-(1H-indole-2-carbonyl)piperidin-3-ol
3-(azocan-1-yl)-N-(furan-3-ylmethyl)-N-methylpropanamide
2-[2,5-dimethyl-1-(pyridin-3-ylmethyl)-1H-pyrrol-3-yl]-1H-1,3-benzodiazole-5-carbonitrile
5-{2-[bis(propan-2-yl)carbamoyl]phenyl}furan-2-carboxamide
2-(ethanesulfonyl)-7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinoline
propan-2-yl 2-chloro-5-(6-oxo-1,6-dihydropyridazine-3-amido)benzoate
8-fluoro-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}quinoline-2-carboxamide
2-[(2,3-difluoro-4-methoxyphenyl)formamido]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
3-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
4-[1-(2-hydroxybutyl)-5-(2-methoxypropan-2-yl)-1H-1,2,4-triazol-3-yl]benzamide
1-cyclopentyl-4-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]-1,4-diazepane
1-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-4-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[3-(pyrrolidin-1-yl)propyl]-1,4-diazepane
6-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-oxo-1,4-dihydropyridine-3-carboxamide
4-[1-(4-chlorophenyl)cyclobutanecarbonyl]-1,4-oxazepan-6-ol
3-cyclopentyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
N-[(2,3-difluorophenyl)methyl]-4-(ethylamino)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[(3R,4S)-1-(4-cyclopentylpyrimidin-2-yl)-4-cyclopropylpyrrolidin-3-yl]-2-hydroxyacetamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-5-phenyl-1,2-oxazole-3-carboxamide
5-(2-fluorophenyl)-N-[1-(1-propyl-1H-1,2,4-triazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(3-chloro-5-methoxybenzoyl)-2-(pyrrolidine-1-carbonyl)piperazine
methyl 4-({2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}sulfonyl)benzoate
N-[2-(4-fluorophenyl)ethyl]-1,3-dimethyl-2,6-dioxo-N-(pyridin-3-ylmethyl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-(furan-2-yl)-N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)propanamide
3-[1-(5-amino-1H-pyrazole-3-carbonyl)piperidin-4-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(1R,3S)-3-(2-aminoethoxy)-7-[(4-phenyl-1,3-thiazol-2-yl)methyl]-7-azaspiro[3.5]nonan-1-ol
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(1-phenoxypropan-2-yl)piperidine
2-[4-methyl-6-(pyridin-3-yl)pyrimidin-2-yl]phenol
N-(2-methoxyethyl)-1-methyl-3-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
5-chloro-N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-methyl-1-benzothiophene-2-sulfonamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-(4-fluorophenoxymethyl)-4-hydroxypyrimidine-5-carboxamide
N-[3-(4-methylpiperazin-1-yl)propyl]-3-phenyl-1H-pyrazole-4-carboxamide
2-[(2S,4S)-2-(diethylcarbamoyl)-4-(2-methyl-1,3-thiazole-4-amido)pyrrolidin-1-yl]acetic acid
1-{2-[(5-tert-butyl-1,3,4-oxadiazol-2-yl)amino]ethyl}imidazolidin-2-one