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N3-butyl-1-(furan-2-ylmethyl)-N5-[(3-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3-[(4-fluorophenyl)methoxy]azetidine
10-methoxy-5-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
{2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}urea
N-(3-methoxyphenyl)-2-[4-(5-methyl-1,2-oxazole-3-carbonyl)morpholin-3-yl]acetamide
2-methyl-N-{2-methyl-3-[(1,3-thiazol-2-yl)carbamoyl]phenyl}-1H-imidazole-4-carboxamide
6-{4-[1-(dimethylamino)ethyl]piperidin-1-yl}-N4-methylpyrimidine-2,4-diamine
1-{3-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]propyl}piperidin-2-one
2-{2-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]phenyl}-5-methyl-1,3,4-oxadiazole
2-[5-(methoxymethyl)furan-2-yl]-1H-1,3-benzodiazole
8-[2-(3,4-difluorophenyl)acetyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{2-[(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]ethyl}acetamide
4-[1-(1H-indole-5-carbonyl)piperidin-3-yl]benzoic acid
N-(4-fluorophenyl)-1-[3-(pyridin-3-yl)propanoyl]piperazine-2-carboxamide
1-(3-{[(furan-2-ylmethyl)amino]methyl}pyridin-2-yl)piperidin-3-ol
N-cyclopentyl-N'-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}butanediamide
4-benzyl-3-ethyl-1-(5-methylpyridine-3-carbonyl)-1,4-diazepan-5-one
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-methyl-N-(thiophen-3-ylmethyl)acetamide
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-[3-(methylsulfanyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{2-[3-methyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,3-benzodiazole
N,N-dimethyl-2-phenyl-7-(1H-pyrazole-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
8-({2-ethyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-[(3-methoxyphenyl)methyl]-4-[2-(thiophen-2-yl)acetyl]-1,4-diazepan-2-one
N-[(3,4-difluorophenyl)methyl]-3-[1-(2-methylfuran-3-carbonyl)piperidin-3-yl]propanamide
2-{9-[(2-fluoro-5-methoxyphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
4-methyl-3-[3-(morpholin-4-ylmethyl)phenyl]benzoic acid
N,2,2-trimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-(thiophen-2-yl)cyclopropane-1-carboxamide
(2S,4R)-4-amino-1-(1,6-dimethyl-1H-indole-2-carbonyl)-N-ethylpyrrolidine-2-carboxamide
(3S,4S)-1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-(prop-2-en-1-yl)-9-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
3-methyl-2-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]pyridine
N-(2,3-dihydro-1H-inden-2-yl)-4-(hydroxymethyl)pyridine-2-carboxamide
3-{1-[(2,4,6-trimethoxyphenyl)methyl]piperidin-2-yl}propanoic acid
2-(1H-1,3-benzodiazol-2-ylmethoxy)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
N-[(3S,4R)-1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
3-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyridine
2-[3-(dimethylamino)phenyl]-N,N-dimethylbenzamide
3-[1-(adamantan-1-yl)piperidin-4-yl]-1-(4-ethylpiperazin-1-yl)propan-1-one
5-{4-[3-(3,4-dimethyl-1H-pyrazol-5-yl)propanoyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
3-{4-[3-(dimethylamino)phenyl]-3,5-dimethyl-1H-pyrazol-1-yl}propanamide
ethyl 4-[(4-methoxyphenyl)methyl]-1-[3-(2-methoxyphenyl)propanoyl]piperidine-4-carboxylate
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methylthiophene-3-carboxamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl){[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-methyl-4-[3-(trifluoromethyl)phenyl]-1H-imidazole
3-[1-(1-cyclopropylethyl)-3-methyl-1H-pyrazol-5-yl]-1-methyl-1-[2-(phenylsulfanyl)ethyl]urea
(1S,5R)-6-(2-methoxyethyl)-3-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)cyclopropanamine
1-[(2-chloro-6-fluorophenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
7-[2-(benzyloxy)ethyl]pyrazolo[1,5-a]pyridine
1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-hydroxypropan-1-one