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N-cyclopentyl-2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoacetamide
1-[(4-methyl-1H-imidazol-5-yl)methyl]-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-[(2-fluorophenyl)methyl]-N-methyl-N-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
1-[3-(dimethylamino)phenyl]-3-methyl-3-[2-(methylsulfanyl)ethyl]urea
methyl({[2-(propan-2-yl)pyrimidin-4-yl]methyl})[1-(pyridin-2-yl)ethyl]amine
1-[1-(3-phenylbutyl)azetidin-3-yl]piperidine
3-{[(3S,4R)-3-acetamido-4-(propan-2-yl)pyrrolidin-1-yl]sulfonyl}-N-methylbenzamide
1-[6-(cyclopentylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-N,N-dimethylpyrrolidin-3-amine
methyl({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl})(quinolin-4-ylmethyl)amine
dimethyl(2-{2-[1-(quinoxaline-6-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3,3-dimethylbutyl)piperidine
N-({1-[(3S,5S)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}methyl)-N-methylpiperidine-1-carboxamide
N-(5-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decane-7-carbonyl}-1,3-thiazol-2-yl)acetamide
1-(1-methyl-1H-pyrazole-3-carbonyl)-2-(2-phenylethyl)piperidine
1-(2-{1-[4-(1H-imidazol-1-yl)butanoyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
methyl 3-{2-oxo-4-[2-(pyridin-3-yl)acetyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl}propanoate
N-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
(4aS,7aR)-1-[(2-ethylphenyl)methyl]-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{7-methylthieno[3,2-d]pyrimidin-4-yl}azepan-3-amine
5-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2-dihydropyridin-2-one
1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-ethoxyethan-1-one
methyl 2-chloro-4-[({2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}carbamoyl)amino]benzoate
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyridine
4-(naphthalen-1-yl)-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-3-fluoroimidazo[1,2-a]pyridine
5-(4-{[3-(hydroxymethyl)-3-methylpiperidin-1-yl]methyl}phenoxymethyl)furan-2-carboxylic acid
4-[2-(pyridin-2-yl)ethyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{5-[2-(furan-2-yl)azepane-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
3-(2-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
2-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]quinoline
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,5-dimethyl-1,3-oxazole-4-carboxamide
(4aS,8aR)-6-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-(2-{2-methyl-1-azatricyclo[6.3.1.04,12]dodeca-2,4,6,8(12)-tetraen-3-yl}ethyl)-1-(1H-1,2,3,4-tetrazol-5-yl)urea
5-chloro-N,15-dimethyl-13-oxo-N-(oxolan-3-yl)-9-phenyl-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
2-[2-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-3,4-dihydroquinazolin-4-one
3-methyl-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(2-methoxyethyl)morpholine
(1S,6R)-9-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
6-(6-hydroxy-1,4-oxazepane-4-carbonyl)-3,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-[2-(3,4-dichlorophenyl)morpholin-4-yl]-N-ethylpropanamide
3-[3-(2-ethyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1-[(5-ethylpyridin-2-yl)methyl]-1-methylurea
methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})[1-(pyridin-2-yl)propan-2-yl]amine
N-({7-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(phenylsulfanyl)acetamide
8-cyclopropanecarbonyl-2-(2-fluorobenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N,N,2,2,3-pentamethyl-3-{3-[(3-methylphenyl)methyl]-1,2,4-oxadiazol-5-yl}cyclopentane-1-carboxamide
ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)(thiophen-3-ylmethyl)amine
8-butanoyl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
8-(5-ethylthiophene-3-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one