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N-[2-(diethylamino)-2-(furan-2-yl)ethyl]-1-methylpiperidin-4-amine
2-{[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]amino}-N-(pyrazin-2-yl)acetamide
N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-3-(thiophen-3-yl)propanamide
N-benzyl-N-(3-hydroxy-2-methylpropyl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-(3-cyano-4-methoxyphenyl)-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
1-{5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl}-4-(pyridin-4-yl)-1,4-diazepane
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methylcyclopropanecarbonyl)piperidine
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl)({5-[(oxolan-2-ylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)amine
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]-2,3-dihydro-1H-indene-2-carboxamide
1-[3-({[2-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-[2-(4-chlorophenyl)ethyl]-N-(2-hydroxyethyl)-6-oxo-N-propylpiperidine-3-carboxamide
2-(4-methoxyphenyl)-7-methyl-3-(thiomorpholin-4-ylmethyl)quinoline
N-{3-[2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)acetamido]phenyl}-3-phenylpropanamide
1-(2-hydroxyethyl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}piperidine-4-carboxamide
5-{[(2,6-dimethylquinolin-4-yl)formamido]methyl}thiophene-2-carboxylic acid
{[2-(4-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}(thiophen-2-ylmethyl)amine
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
N-(4-cyanophenyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
3-{[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-4-propyl-4H-1,2,4-triazole
8-(2-methoxypyridine-3-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{2-[(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)formamido]ethyl}pyridine-3-carboxamide
3-[4-(1-benzothiophen-3-yl)-1H-pyrazol-1-yl]propanamide
3-[(3R,4S)-1-[2-(2-fluorophenyl)acetyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-methyl-4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(2H-1,3-benzodioxol-5-yl)-5-(cyclopropylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
2-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,3'-piperidine]-1'-yl}pyridine-3-carbonitrile
3-{[(2-methoxyethyl)[(2-methylphenyl)methyl]amino]methyl}-1-methyl-1,2-dihydroquinolin-2-one
1-(ethanesulfonyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-(isoquinolin-5-ylmethyl)-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
(3R,4R)-1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-[2-(pyridin-2-yl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
4-[(4-benzoylpiperazin-1-yl)methyl]-2,6-dimethylphenyl acetate
6-(4-chlorophenyl)-N-[1-(pyridin-3-yl)propan-2-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{[1-(1-carbamoylethyl)piperidin-4-yl]oxy}-3-chloro-N-[2-(dimethylamino)ethyl]benzamide
2-(butylsulfanyl)-N4-(pyridin-3-ylmethyl)pyrimidine-4,6-diamine
3-({[(dimethylcarbamoyl)methyl]carbamoyl}methyl)-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
[1-(2,6-dimethylpyrimidine-4-carbonyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
1-methyl-8-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(1,4-dioxan-2-ylmethyl)-5-[(2-methyl-1H-imidazol-1-yl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
3-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1-(2,3-dihydro-1H-inden-4-yl)-3-methylurea
N-{1-[(4-fluorophenyl)methyl]-7-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
(1R,3S)-3-({1-[(2-chlorophenyl)methyl]piperidin-4-yl}carbamoyl)cyclopentane-1-carboxylic acid
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-4,5,6,7-tetrahydro-2-benzothiophene-1-carboxamide
2-methyl-6-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
1-(4-methyl-2-{[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]amino}pyrimidin-5-yl)ethan-1-one
1-{[4-(1H-pyrazol-4-yl)phenyl]methyl}piperidine
2-{4-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
4-{4-[2-(3-chlorophenyl)-1H-imidazol-1-yl]benzoyl}morpholine