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3-[N-benzyl-3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamido]propanamide
3-[4-(3,4-dichlorophenyl)piperazine-1-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
1-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-(morpholin-3-yl)ethan-1-one
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-3-(dimethyl-1,2-oxazol-4-yl)propanamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
3-(4-phenyl-1,4-diazepane-1-carbonyl)piperidine-1-carboxamide
N-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
(4-{[methyl({[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl})amino]methyl}oxan-4-yl)methanol
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)azepane
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(morpholin-4-yl)ethane-1,2-dione
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-(4-methoxyphenyl)cyclopentane-1-carboxamide
(2S,4R)-4-amino-1-[(5-cyclopentylthiophen-2-yl)methyl]-N-methylpyrrolidine-2-carboxamide
4-chloro-N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-2-hydroxybenzamide
(1S,5R)-3-(oxan-4-yl)-6-[3-(1H-pyrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
1-[2-(4-chlorophenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]azepane
5-({3-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)pyrimidine
3-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]-4-(pyridin-2-ylmethyl)piperazin-2-one
(3aS,6aS)-2-cyclobutanecarbonyl-5-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyrimidine
3-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-N-(pyridin-3-yl)propanamide
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-pyrazol-4-yl)ethyl]amine
1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-phenylpropan-1-one
3-benzyl-8-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-{[(2,5-difluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
propan-2-yl N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)carbamate
1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-(3-methoxyphenoxymethyl)piperidine
2-[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-2-yl]pyridine
N-butyl-N,5-dimethyl-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-(hydroxymethyl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1H-1,3-benzodiazole-5-carboxamide
4-{2-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethyl}morpholine
[3-(3-methylbut-2-en-1-yl)-1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]methanol
1-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carbonyl)piperidin-3-ol
N-(1-hydroxy-2-methylpropan-2-yl)-3-(2-methylphenyl)-3-phenylpropanamide
2-{2-[1-(1-benzothiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-(3-aminopropyl)-3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)propanamide
(3S,4R)-1-(2-amino-2-methylpropanoyl)-4-phenylpyrrolidine-3-carboxylic acid
(1S,5R)-3-methyl-6-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
2-(dimethyl-1,2-oxazol-4-yl)-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]acetamide
6-[({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)amino]pyridine-2-carbonitrile
4-(4-{1-[(4-methylpyridin-2-yl)methyl]-1H-1,2,3-triazol-4-yl}phenyl)but-3-yn-1-ol
N-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
N-(5-chloro-2-ethyl-3-methyl-1-benzofuran-7-yl)-3-oxopiperazine-1-carboxamide
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrazine
N-[(5-fluoro-1H-indol-2-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}cyclobutanecarboxamide
2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(2-hydroxypropyl)acetamide
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-N-methyl-N-(2-phenylethyl)piperidin-3-amine
N-benzyl-N-(2-hydroxyethyl)-15-methyl-13-oxo-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-3-[(2-methylbutyl)amino]-5-(pyrrolidine-1-sulfonyl)benzamide
N-[(1R,2S)-2-phenylcyclopropyl]-2-(4-propanoylphenoxy)acetamide