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2-{1-[1-(methoxymethyl)cyclobutanecarbonyl]pyrrolidin-2-yl}-6-methyl-1H-1,3-benzodiazole
methyl 1-(3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanoyl)piperidine-2-carboxylate
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(thiophene-3-carbonyl)pyrrolidin-3-yl]methanol
7-(furan-2-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-{2-[2-(1-phenylethyl)-1H-imidazol-1-yl]ethyl}-1,3-oxazinan-2-one
methyl 2-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}piperidine-1-carboxylate
9-(3-chloro-4-methylbenzoyl)-3,9-diazaspiro[5.6]dodecane
N-(1H-indazol-5-yl)-4-methoxy-4-(prop-2-en-1-yl)piperidine-1-carboxamide
4-methyl-2-phenyl-1-(1H-1,2,3-triazole-5-carbonyl)piperazine
(1S,5R)-6-(cyclopropylmethyl)-3-[3-(pyridin-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidin-3-yl)piperidine
(1R,5R)-6-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-{imidazo[1,2-a]pyridin-2-yl}-N-[1-(1H-indol-2-yl)ethyl]-N-methylpropanamide
3-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}pyridin-2-ol
1-[2-(1-benzothiophen-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidine-3-carboxamide
(1R,7S)-N-methyl-4-oxo-3-[4-(propan-2-yl)phenyl]-N-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-{2-[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
{3-[(3-ethyl-1H-pyrazol-5-yl)methyl]-9-[3-(methylsulfanyl)propyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
5-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-butyl-3-[(3-hydroxypiperidin-1-yl)methyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide
2-[(2-chlorophenyl)methyl]-4-[2,2-dimethyl-3-(morpholin-4-yl)propyl]morpholine
1-[3-(morpholin-4-yl)propyl]-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
2-[3-(1H-imidazol-1-yl)propyl]-9-(3,3,3-trifluoro-2-methylpropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(3R,4S)-1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
1-cyclohexyl-4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
7-(1-benzofuran-5-carbonyl)-2-(dimethylamino)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-phenyl-1H-imidazol-5-yl}quinolin-8-ol
3-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-methylpiperidine
1-(2,4-dimethoxyphenyl)-2-(4-methanesulfonylphenyl)-1H-imidazole
[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl](methyl){[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
5-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylic acid
6-(4-methyl-1,4-diazepan-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-(2-methylpropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-methoxy-4-({[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
1-methyl-4-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-1,4-diazepane
1-[(3-fluorophenyl)methyl]-4-[4-(furan-2-yl)benzoyl]piperazine
N-cyclopropyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
2-{[5-(3-cyanophenyl)-4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-1,2-oxazole-3-carboxamide
4-[4-amino-6-(benzylamino)-1,3,5-triazin-2-yl]benzonitrile
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide
3-{imidazo[1,2-a]pyridin-2-ylmethyl}-3H,4H-pyrido[2,3-d]pyrimidin-4-one
4-[1-(2-ethoxyethyl)piperidin-3-yl]benzoic acid
5-{5-[1-(cyclohexylmethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
2-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
3-(1H-pyrazol-1-ylmethyl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}benzamide
(3S,4S)-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-4-methylpiperidine-3,4-diol