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2-{4-[2-amino-3-cyano-6-(propan-2-yl)pyridin-4-yl]-2-chlorophenoxy}acetamide
6-[1-(1-ethylpyrrolidine-3-carbonyl)piperidin-4-yl]pyrimidin-4-ol
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
3-(3-chloro-1,2-oxazol-5-yl)-N-(1H-indol-4-ylmethyl)propanamide
1-(5-{[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-[2-(methylamino)ethyl]-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
1-[1-(furan-2-carbonyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
2-(5-{1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
5-(hydroxymethyl)-2-methyl-4-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}pyridin-3-ol
N-(dicyclopropylmethyl)-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
N-methyl-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}acetamide
1-benzyl-3-[2-(3-methoxypyrrolidin-1-yl)-2-oxoethyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
1-methyl-6-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
N-[(3S,4R)-1-(1H-indole-6-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
3-{[2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl](methyl)amino}-1λ6-thiolane-1,1-dione
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
7-[3-(1H-indol-3-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]-2-methyl-1,4-diazepan-5-one
4-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-oxobutanamide
1-methyl-3-[2-(methylsulfanyl)ethyl]-5-(5-methylthiophen-2-yl)-1H-1,2,4-triazole
1-(3-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-oxopropyl)-1,2-dihydropyridin-2-one
2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-(2,3-dihydro-1,4-benzodioxin-6-yl)acetic acid
N,N-diethyl-2-(2-ethylpyrimidin-5-yl)-5,7-dimethylquinoline-4-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]oxolane-3-carboxamide
2-[(3-carbamoyl-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]pyridine-3-carboxylic acid
N-[2-(3,5-dimethylphenoxy)ethyl]-N-methyl-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
2-(2,5-dioxoimidazolidin-4-yl)-N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}acetamide
2-methyl-4-(2-methylphenyl)-1-(pyridin-4-ylmethyl)piperazine
N'-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]ethanediamide
2-(2-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)-1,2-oxazinane
N-benzyl-3-{[(2-hydroxypropyl)(methyl)amino]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
3-methyl-3-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-1-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
3-(3-fluoro-4-methoxybenzoyl)-1-(oxan-4-yl)piperidine
(3aS,6aS)-2-(ethanesulfonyl)-5-(1,3-thiazol-4-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-N-(4-{[1-(3-methylpyridin-2-yl)propan-2-yl]carbamoyl}phenyl)furan-3-carboxamide
1-[4-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-(pyridin-3-yloxy)ethan-1-one
ethyl (2S)-2-[4-(4-ethoxy-3-methylphenyl)butanamido]propanoate
3-{1-[2-(4-chlorophenoxy)acetyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
5-hydroxy-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]pyridine-2-carboxamide
2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
3-[(2-fluorophenyl)formamido]-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)propanamide
methyl (2S)-2-{[2-(2,3-difluorophenoxymethyl)-1,3-oxazol-4-yl]formamido}-3-methylbutanoate
4-[(4-hydroxyphenyl)methyl]-1-(oxan-4-ylmethyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-[3-(methylsulfanyl)propyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-ethyl-5-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
ethyl 1-[1-(ethoxycarbonyl)piperidin-4-yl]-4-(2-methoxyethyl)piperidine-4-carboxylate
(1s,4s)-4-{4-[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
1-[4-(2-{[2-(2-methoxyethyl)piperidin-1-yl]methyl}-8-methylquinazolin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide